# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA854490 | B | Activity against DYRK2 at 10 uM in the presence of 100 uM ATP relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
2. | ALA1806166 | B | Inhibition of DYRK2 assessed as residual enzyme activity at 10 uM | 1 | single protein format | Scientific Literature | |||
3. | ALA1664065 | B | Inhibition of DYRK2 at 1 uM | 2 | single protein format | Scientific Literature | |||
4. | ALA2014114 | B | Inhibition of human N-terminal GST-tagged DYRK2 expressed in baculovirus using DYRKtide-F as substrate assessed as inhibition of [33P] incorporation into substrate using [gamma33P]ATP after 10 mins by liquid scintillation counting | Homo sapiens | 18 | assay format | Scientific Literature | ||
5. | ALA2015848 | B | Inhibition of DYRK2 assessed as residual activity at 1 uM relative to control | 1 | single protein format | Scientific Literature | |||
6. | ALA2014920 | B | Inhibition of DYRK2 at 10 uM | 1 | single protein format | Scientific Literature | |||
7. | ALA2015537 | B | Inhibition of DYRK2 | 2 | single protein format | Scientific Literature | |||
8. | ALA2015004 | B | Inhibition of DYRK2 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
9. | ALA1805100 | B | Inhibition of human recombinant GST-tagged DYRK2 using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation counting | Homo sapiens | 39 | single protein format | Scientific Literature | ||
10. | ALA1805108 | B | Inhibition of human recombinant GST-tagged DYRK2 using KISGRLSPIMTEQ as substrate and [gamma32]-ATP at 10 uM after 30 mins by scintillation counting | Homo sapiens | 3 | single protein format | Scientific Literature | ||
11. | ALA1805116 | B | Inhibition of recombinant DYRK2-mediated SR 9G8 protein phosphorylation at 10 uM after 30 mins by SDS-PAGE followed by autoradiography | 1 | single protein format | Scientific Literature | |||
12. | ALA1827233 | B | Activity of DYRK2 kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
13. | ALA1962040 | B | GSK_PKIS: DYRK2 mean inhibition at 0.1 uM [Nanosyn] | 366 | single protein format | GSK Published Kinase Inhibitor Set | |||
14. | ALA1962041 | B | GSK_PKIS: DYRK2 mean inhibition at 1 uM [Nanosyn] | 366 | single protein format | GSK Published Kinase Inhibitor Set | |||
15. | ALA922814 | B | Activity of human DYRK2 kinase at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
16. | ALA973719 | B | Inhibition of human DYRK2 kinase assessed as residual enzyme activity at 0.1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
17. | ALA950866 | B | Inhibition of human DYRK2 at 10 uM | 1 | single protein format | Scientific Literature | |||
18. | ALA1003336 | B | Inhibition of DYRK2 at 1 uM relative to control | 3 | single protein format | Scientific Literature | |||
19. | ALA954302 | B | Inhibition of human DYRK2 at 10 uM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
20. | ALA1061748 | B | Inhibition of DYRK2 at 1 uM | 1 | single protein format | Scientific Literature |