| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA856393 | B | Percent residual activity, relative to control, of ERK8 at 1 uM concentration of inhibitor in presence of 5 uM ATP | Homo sapiens | 2 | ALA1137240 | single protein format | Scientific Literature | |
| 2. | ALA945011 | B | Residual activity of ERK8 at 10 uM relative to control | 3 | ALA1141471 | single protein format | Scientific Literature | ||
| 3. | ALA949029 | B | Inhibition of ERK8 at 10 uM | 1 | ALA1143865 | single protein format | Scientific Literature | ||
| 4. | ALA950854 | B | Inhibition of ERK8 at 10 uM | 1 | ALA1137681 | single protein format | Scientific Literature | ||
| 5. | ALA1000625 | B | Inhibition of ERK8 at 1 uM relative to control | 3 | ALA1136991 | single protein format | Scientific Literature | ||
| 6. | ALA983618 | B | Inhibition of ERK8 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 7. | ALA1061960 | B | Percentage ERK8 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
| 8. | ALA1060193 | B | Binding constant for ERK8 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 9. | ALA1061212 | B | Percentage ERK8 activity remaining in the presence of 0.01uM inhibitor | Homo sapiens | 3 | ALA1150976 | single protein format | Scientific Literature | |
| 10. | ALA1061213 | B | Percentage ERK8 activity remaining in the presence of 3uM inhibitor | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
| 11. | ALA1060116 | B | Percentage ERK8 activity remaining in the presence of 25uM inhibitor | Homo sapiens | 2 | ALA1150976 | single protein format | Scientific Literature | |
| 12. | ALA1060117 | B | Percentage ERK8 activity remaining in the presence of 2uM inhibitor | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
| 13. | ALA1052076 | B | Percentage ERK8 activity remaining in the presence of 10uM inhibitor | Homo sapiens | 24 | ALA1150976 | single protein format | Scientific Literature | |
| 14. | ALA1062012 | B | Percentage ERK8 activity remaining in the presence of 1uM inhibitor | Homo sapiens | 33 | ALA1150976 | single protein format | Scientific Literature | |
| 15. | ALA1057674 | B | Inhibition of ERK8 assessed as remaining enzyme activity at 1 uM relative to DMSO | 1 | ALA1154183 | single protein format | Scientific Literature | ||
| 16. | ALA1047336 | B | Inhibition of ERK8 assessed as residual enzyme activity at 10 uM relative to untreated control | 4 | ALA1154186 | single protein format | Scientific Literature | ||
| 17. | ALA1053724 | B | Inhibition of ERK8 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 18. | ALA1046789 | B | Inhibition of ERK8 assessed as remaining enzyme activity at 3 uM relative to DMSO | 1 | ALA1154183 | single protein format | Scientific Literature | ||
| 19. | ALA1048078 | B | Inhibition of ERK8 assessed as residual activity at 10 uM by Cherenkov counting relative to control in presence of 5 uM ATP | 2 | ALA1155278 | single protein format | Scientific Literature | ||
| 20. | ALA1048100 | B | Inhibition of ERK8 assessed as residual activity at 0.1 uM by Cherenkov counting relative to control in presence of 5 uM ATP | 2 | ALA1155278 | single protein format | Scientific Literature |
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