# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA856397 | B | Percent residual activity, relative to control, of MNK1 at 1 uM concentration of inhibitor in presence of 50 uM ATP | Homo sapiens | 2 | ALA1137240 | single protein format | Scientific Literature | |
2. | ALA904792 | B | Inhibition of MNK1 | Homo sapiens | 4 | ALA1143661 | single protein format | Scientific Literature | |
3. | ALA922897 | B | Inhibition of MNK1 | 1 | ALA1140654 | single protein format | Scientific Literature | ||
4. | ALA950812 | B | Inhibition of MNK1 at 10 uM | 1 | ALA1137681 | single protein format | Scientific Literature | ||
5. | ALA950855 | B | Inhibition of MNK1 at 10 uM | 1 | ALA1137681 | single protein format | Scientific Literature | ||
6. | ALA999773 | B | Binding affinity to human MKNK1 at 5 uM | Homo sapiens | 2 | ALA1136966 | single protein format | Scientific Literature | |
7. | ALA1000640 | B | Inhibition of MNK1 at 1 uM relative to control | 3 | ALA1136991 | single protein format | Scientific Literature | ||
8. | ALA987192 | B | Inhibition of MKNK1 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
9. | ALA1062763 | B | Percentage MNK1 activity remaining in the presence of 3uM inhibitor | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
10. | ALA1052105 | B | Percentage MNK1 activity remaining in the presence of 25uM inhibitor | Homo sapiens | 2 | ALA1150976 | single protein format | Scientific Literature | |
11. | ALA1061970 | B | Percentage MNK1 activity remaining in the presence of 10uM inhibitor | Homo sapiens | 24 | ALA1150976 | single protein format | Scientific Literature | |
12. | ALA1063758 | B | Percentage MNK1 activity remaining in the presence of 0.01uM inhibitor | Homo sapiens | 3 | ALA1150976 | single protein format | Scientific Literature | |
13. | ALA1063759 | B | Percentage MNK1 activity remaining in the presence of 1uM inhibitor | Homo sapiens | 33 | ALA1150976 | single protein format | Scientific Literature | |
14. | ALA1063760 | B | Percentage MNK1 activity remaining in the presence of 2uM inhibitor | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
15. | ALA1063804 | B | Binding constant for full-length MKNK1 | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
16. | ALA1062792 | B | Inhibition of MNK1 in the presence of 50uM ATP | Homo sapiens | 2 | ALA1150976 | single protein format | Scientific Literature | |
17. | ALA1060206 | B | Percentage MNK1 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
18. | ALA1060295 | B | Inhibition of MNK1 assessed as remaining enzyme activity at 1 uM relative to DMSO | 1 | ALA1154183 | single protein format | Scientific Literature | ||
19. | ALA1056863 | B | Inhibition of MNK1 assessed as residual enzyme activity at 10 uM relative to untreated control | 4 | ALA1154186 | single protein format | Scientific Literature | ||
20. | ALA1047452 | B | Inhibition of MKNK1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature |