| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1004483 | B | Binding affinity to human recombinant PIM3 expressed in Escherichia coli assessed as thermal shift by differential scanning fluorimetry | Homo sapiens | 7 | ALA1140872 | assay format | Scientific Literature | |
| 2. | ALA945701 | B | Inhibition of human PIM3 at 10 uM | 1 | ALA1137681 | single protein format | Scientific Literature | ||
| 3. | ALA1000639 | B | Inhibition of PIM3 at 1 uM relative to control | 3 | ALA1136991 | single protein format | Scientific Literature | ||
| 4. | ALA970287 | B | Inhibition of PIM3 at 10 uM | 1 | ALA1156515 | single protein format | Scientific Literature | ||
| 5. | ALA981741 | B | Inhibition of PIM3 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 6. | ALA1061167 | B | Percentage PIM3 activity remaining in the presence of 2uM inhibitor | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
| 7. | ALA1061168 | B | Percentage PIM3 activity remaining in the presence of 3uM inhibitor | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
| 8. | ALA1061195 | B | Inhibition of PIM3 in the presence of 5uM ATP | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
| 9. | ALA1062887 | B | Inhibition of PIM3 in the presence of 20uM ATP | Homo sapiens | 4 | ALA1150976 | single protein format | Scientific Literature | |
| 10. | ALA1051340 | B | Binding constant for PIM3 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 11. | ALA1051343 | B | Percentage PIM3 activity remaining in the presence of 10uM inhibitor | Homo sapiens | 24 | ALA1150976 | single protein format | Scientific Literature | |
| 12. | ALA1061911 | B | Percentage PIM3 activity remaining in the presence of 0.01uM inhibitor | Homo sapiens | 3 | ALA1150976 | single protein format | Scientific Literature | |
| 13. | ALA1061912 | B | Percentage PIM3 activity remaining in the presence of 1uM inhibitor | Homo sapiens | 33 | ALA1150976 | single protein format | Scientific Literature | |
| 14. | ALA1051300 | B | Percentage PIM3 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
| 15. | ALA1051328 | B | Inhibition of PIM3 in the presence of 100uM ATP | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
| 16. | ALA1060258 | B | Percentage PIM3 activity remaining in the presence of 25uM inhibitor | Homo sapiens | 2 | ALA1150976 | single protein format | Scientific Literature | |
| 17. | ALA1059320 | B | Inhibition of human PIM3 by scintillation counting | Homo sapiens | 12 | ALA1154637 | single protein format | Scientific Literature | |
| 18. | ALA1056912 | B | Inhibition of PIM3 assessed as remaining enzyme activity at 3 uM relative to DMSO | 1 | ALA1154183 | single protein format | Scientific Literature | ||
| 19. | ALA1055336 | B | Inhibition of PIM3 assessed as remaining enzyme activity at 1 uM relative to DMSO | 1 | ALA1154183 | single protein format | Scientific Literature | ||
| 20. | ALA1057615 | B | Inhibition of Pim-3 assessed as residual enzyme activity at 10 uM relative to untreated control | 19 | ALA1154186 | single protein format | Scientific Literature |
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