| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA904249 | B | Inhibition of GST-p300 HAT assessed as histone acetylation | Homo sapiens | 8 | ALA1142987 | single protein format | Scientific Literature | |
| 2. | ALA904259 | B | Activity of GST-p300 HAT assessed as HAT activity at 5 uM | Homo sapiens | 1 | ALA1142987 | single protein format | Scientific Literature | |
| 3. | ALA904260 | B | Activity of GST-p300 HAT assessed as HAT activity at 21 uM | Homo sapiens | 1 | ALA1142987 | single protein format | Scientific Literature | |
| 4. | ALA904262 | B | Inhibition of GST-p300 HAT expressed in bacteria assessed as histone acetylation | 1 | ALA1142987 | assay format | Scientific Literature | ||
| 5. | ALA904261 | B | Inhibition of full length GST-p300 expressed in Sf9 cells assessed as histone acetylation | Homo sapiens | 1 | ALA1142987 | cell-based format | Scientific Literature | |
| 6. | ALA1006960 | B | Inhibition of recombinant His-tagged HAT p300 expressed in Sf21-Baculovirus system | 1 | ALA1140879 | assay format | Scientific Literature | ||
| 7. | ALA1006961 | B | Inhibition of HAT p300 | 1 | ALA1140879 | single protein format | Scientific Literature | ||
| 8. | ALA1006964 | B | Inhibition of GST-fused recombinant HAT p300 expressed in Escherichia coli by filter assay | 6 | ALA1140879 | assay format | Scientific Literature | ||
| 9. | ALA1025548 | B | Inhibition of recombinant p300 | 10 | ALA1143309 | single protein format | Scientific Literature | ||
| 10. | ALA1029896 | B | Inhibition of human immunoprecipitated histone acetyltransferase p300 in U937 cell nuclear extracts assessed as remaining enzyme activity at 50 uM | Homo sapiens | 10 | ALA1136851 | cell-based format | Scientific Literature | |
| 11. | ALA1021609 | B | Inhibition of HAT p300 catalytic domain R1627K mutant expressed in Escherichia coli BL21 up to 100 uM by fluorography/autoradiography assay | Homo sapiens | 1 | ALA1139360 | assay format | Scientific Literature | |
| 12. | ALA1021610 | B | Inhibition of HAT p300 catalytic domain G1626A mutant expressed in Escherichia coli BL21 up to 100 uM by fluorography/autoradiography assay | Homo sapiens | 1 | ALA1139360 | assay format | Scientific Literature | |
| 13. | ALA1021611 | B | Inhibition of HAT p300 catalytic domain Y1397F mutant expressed in Escherichia coli BL21 up to 100 uM by fluorography/autoradiography assay | Homo sapiens | 1 | ALA1139360 | assay format | Scientific Literature | |
| 14. | ALA1021612 | B | Inhibition of HAT p300 catalytic domain S1396A mutant expressed in Escherichia coli BL21 up to 100 uM by fluorography/autoradiography assay | Homo sapiens | 1 | ALA1139360 | assay format | Scientific Literature | |
| 15. | ALA1021613 | B | Inhibition of HAT p300 catalytic domain by equilibrium dialysis | 3 | ALA1139360 | single protein format | Scientific Literature | ||
| 16. | ALA1021614 | B | Binding affinity to HAT p300 catalytic domain by isothermal titration calorimetry | 3 | ALA1139360 | single protein format | Scientific Literature | ||
| 17. | ALA1021615 | B | Inhibition of HAT p300 catalytic domain assessed as drug-induced alteration of protein tertiary structure at 2.5 uM by Stern-Volmer plot | 3 | ALA1139360 | single protein format | Scientific Literature | ||
| 18. | ALA1021616 | B | Inhibition of HAT p300 catalytic domain assessed as drug-induced alteration of protein secondary structure by Stern-Volmer plot | 2 | ALA1139360 | single protein format | Scientific Literature | ||
| 19. | ALA1021617 | B | Binding affinity to HAT p300 catalytic domain by fluorometric titration | 3 | ALA1139360 | single protein format | Scientific Literature | ||
| 20. | ALA1021618 | B | Inhibition of HAT p300 catalytic domain activity expressed in Escherichia coli BL21 (DE3) co-transformed with human SirT2 by fluorography/autoradiography assay | 3 | ALA1139360 | assay format | Scientific Literature |
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