| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA904250 | B | Activity of GST-PCAF assessed as HAT activity at 5 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 2. | ALA904251 | B | Activity of GST-PCAF assessed as HAT activity at 21 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA1798475 | B | Increase of human recombinant KAT2B acetylation activity using histone H4 peptide as substrate at 50 uM after 2 hrs | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 4. | ALA1798476 | B | Inhibition of human recombinant KAT2B using histone H4 peptide as substrate at 50 uM after 2 hrs | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 5. | ALA1832997 | B | Binding affinity to PCAF assessed as change in melting temperature at 100 uM by differential scanning fluorimetry | 9 | single protein format | Scientific Literature | |||
| 6. | ALA1938100 | B | Inhibition of human recombinant His-tagged PCAF HAT domain expressed in Escherichia coli BL21(DE3) cells using [14C]Ac-AoA and histone H4 as substrate at 200 uM after 5 mins by scintillation counting | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 7. | ALA1938103 | B | Inhibition of human recombinant His-tagged PCAF HAT domain expressed in Escherichia coli BL21(DE3) cells using [14C]Ac-AoA and histone H4 as substrate after 5 mins by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA1938105 | B | Inhibition of human recombinant His-tagged PCAF HAT domain expressed in Escherichia coli BL21(DE3) cells using [14C]Ac-AoA and histone H4 as substrate at >200 uM after 5 mins by scintillation counting | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 9. | ALA1958936 | B | Binding affinity to PCAF assessed as change in melting temperature at 100 uM by protein stability shift assay | 12 | single protein format | Scientific Literature | |||
| 10. | ALA1959063 | B | Binding affinity to PCAF assessed as change in melting temperature at 10 uM by protein stability shift assay | 6 | single protein format | Scientific Literature | |||
| 11. | ALA900963 | B | Inhibition of PCAF HAT at 50 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA1798494 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli at 50 uM using biotinylated oligopeptide sequences from histone H4 (2-24) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 13. | ALA1798495 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli at 200 uM using biotinylated oligopeptide sequences from histone H4 (2-24) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA1798510 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli using biotinylated oligopeptide sequences from histone H3 (1-21) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 29 | assay format | Scientific Literature | ||
| 15. | ALA1798511 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli using biotinylated oligopeptide sequences from histone H4 (2-24) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 35 | assay format | Scientific Literature | ||
| 16. | ALA1798512 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli at 10 uM using biotinylated oligopeptide sequences from histone H3 (1-21) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA1798513 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli at 25 uM using biotinylated oligopeptide sequences from histone H3 (1-21) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 18. | ALA1798514 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli at 50 uM using biotinylated oligopeptide sequences from histone H3 (1-21) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 7 | assay format | Scientific Literature | ||
| 19. | ALA1798515 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli at 300 uM using biotinylated oligopeptide sequences from histone H3 (1-21) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA1798706 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli using biotinylated oligopeptide sequences from histone H3 (1-21) substrate in presence of 1 mmol/L DTT by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 1 | assay format | Scientific Literature |
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