| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA904250 | B | Activity of GST-PCAF assessed as HAT activity at 5 uM | Homo sapiens | 1 | ALA1142987 | single protein format | Scientific Literature | |
| 2. | ALA904251 | B | Activity of GST-PCAF assessed as HAT activity at 21 uM | Homo sapiens | 1 | ALA1142987 | single protein format | Scientific Literature | |
| 3. | ALA900963 | B | Inhibition of PCAF HAT at 50 uM | Homo sapiens | 1 | ALA1137607 | single protein format | Scientific Literature | |
| 4. | ALA936437 | B | Effect on PCAF in human U937 cells assessed as increase in acetylation activity at 50 uM | Homo sapiens | 1 | ALA1145635 | cell-based format | Scientific Literature | |
| 5. | ALA1006962 | B | Inhibition of HAT PCAF | 1 | ALA1140879 | single protein format | Scientific Literature | ||
| 6. | ALA1006963 | B | Inhibition of GST-fused recombinant HAT PCAF expressed in Escherichia coli by filter assay | 20 | ALA1140879 | assay format | Scientific Literature | ||
| 7. | ALA1001098 | B | Inhibition of human recombinant HAT PCAF | Homo sapiens | 19 | ALA1140889 | single protein format | Scientific Literature | |
| 8. | ALA1025549 | B | Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3) | 9 | ALA1143309 | assay format | Scientific Literature | ||
| 9. | ALA1027324 | B | Inhibition of human GST-fused histone acetyltransferase PCAF in U937 cell nuclear extracts assessed as remaining enzyme activity at 50 uM | Homo sapiens | 10 | ALA1136851 | cell-based format | Scientific Literature | |
| 10. | ALA1021605 | B | Inhibition of HAT PCAF up to 10 uM after 2 mins in absence of acetyl-CoA | 1 | ALA1139360 | single protein format | Scientific Literature | ||
| 11. | ALA1021606 | B | Inhibition of HAT PCAF relative to control | 1 | ALA1139360 | single protein format | Scientific Literature | ||
| 12. | ALA1021607 | B | Inhibition of HAT PCAF up to 40 uM relative to control | 1 | ALA1139360 | single protein format | Scientific Literature | ||
| 13. | ALA1021608 | B | Inhibition of HAT PCAF up to 80 uM relative to control | 1 | ALA1139360 | single protein format | Scientific Literature | ||
| 14. | ALA1047520 | B | Inhibition of human recombinant histone acetyltransferase PCAF assessed as CoA-SH activity preincubated for 15 mins by CPM fluorescent assay | Homo sapiens | 16 | ALA1155178 | single protein format | Scientific Literature | |
| 15. | ALA1219176 | B | Inhibition of human recombinant histone deacetylase PCAF by ELISA | Homo sapiens | 9 | ALA1212875 | single protein format | Scientific Literature | |
| 16. | ALA1219177 | B | Inhibition of human recombinant histone deacetylase PCAF at 1 mM by ELISA | Homo sapiens | 2 | ALA1212875 | single protein format | Scientific Literature | |
| 17. | ALA1219178 | B | Inhibition of histone deacetylase PCAF in human HepG2 cells assessed as decrease in SAHA-induced histone H4 acetylation levels at 30 uM after 24 hrs by Western blotting | Homo sapiens | 2 | ALA1212875 | cell-based format | Scientific Literature | |
| 18. | ALA1219179 | B | Inhibition of histone deacetylase PCAF in human HepG2 cells assessed as decrease in SAHA-induced histone H4 acetylation levels at 60 uM after 24 hrs by Western blotting | Homo sapiens | 2 | ALA1212875 | cell-based format | Scientific Literature | |
| 19. | ALA1798494 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli at 50 uM using biotinylated oligopeptide sequences from histone H4 (2-24) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 4 | ALA1795276 | assay format | Scientific Literature | |
| 20. | ALA1798495 | B | Inhibition of histone acetylase activity of human recombinant PCAF expressed in Escherichia coli at 200 uM using biotinylated oligopeptide sequences from histone H4 (2-24) substrate by In-vitro time-resolved fluorescence immunosorbent acetyltransferase assay | Homo sapiens | 1 | ALA1795276 | assay format | Scientific Literature |
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