# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA904252 | B | Activity of GST-GCN5 assessed as HAT activity at 5 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
2. | ALA904253 | B | Activity of GST-GCN5 assessed as HAT activity at 21 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
3. | ALA1794507 | F | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of GCN5L2: Hit confirmation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504398] | 145 | assay format | PubChem BioAssays | |||
4. | ALA937311 | B | Inhibition of GCN5 in human U937 cells at 50 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
5. | ALA1027323 | B | Inhibition of human histone acetyltransferase GCN5 in U937 cell nuclear extracts assessed as remaining enzyme activity at 50 uM | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
6. | ALA1015489 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.8 mM by Western blot analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
7. | ALA1015490 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.2 mM by Western blot analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
8. | ALA1016346 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.8 mM by Western blot analysis in presence of 100 ng histone H3 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
9. | ALA1016347 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.8 mM by Western blot analysis in presence of 200 ng histone H3 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
10. | ALA1016348 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.8 mM by Western blot analysis in presence of increased concentration of acetyl-CoA | Homo sapiens | 1 | single protein format | Scientific Literature | ||
11. | ALA1016349 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.2 mM by Western blot analysis in presence of histone H3 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
12. | ALA1738606 | F | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of GCN5L2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504398] | Homo sapiens | 13,828 | assay format | PubChem BioAssays | ||
13. | ALA3118017 | B | Inhibition of human recombinant histone acetyltransferase GCN5 assessed as acetylation of histone H3 at 0.15 to 0.6 mM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
14. | ALA3223010 | B | Inhibition of KAT2A (362 to 837) (unknown origin) using biotinylated histone H3 as substrate after 10 mins by TR-FRET analysis relative to control | Homo sapiens | 7 | single protein format | Scientific Literature | ||
15. | ALA3223011 | B | Inhibition of KAT2A (362 to 837) (unknown origin) using biotinylated histone H3 as substrate at 50 uM after 10 mins by TR-FRET analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
16. | ALA3391520 | B | Inhibition of human GCN5 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
17. | ALA3383425 | B | Inhibition of human GCN5 by BROMOscan assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
18. | ALA3424831 | B | Inhibition of recombinant GCN5 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
19. | ALA3591397 | B | Binding affinity to KAT2A in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
20. | ALA3626890 | B | Inhibition of recombinant human KAT2A using biotinylated histone H3 (1 to 21 amino acid residues) as substrate at 50 uM preincubated for 10 mins followed by acetyl-CoA addition measured after 10 mins by time resolved fluorescence assay | Homo sapiens | 28 | single protein format | Scientific Literature |