| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA904252 | B | Activity of GST-GCN5 assessed as HAT activity at 5 uM | Homo sapiens | 1 | ALA1142987 | single protein format | Scientific Literature | |
| 2. | ALA904253 | B | Activity of GST-GCN5 assessed as HAT activity at 21 uM | Homo sapiens | 1 | ALA1142987 | single protein format | Scientific Literature | |
| 3. | ALA937311 | B | Inhibition of GCN5 in human U937 cells at 50 uM | Homo sapiens | 1 | ALA1145635 | cell-based format | Scientific Literature | |
| 4. | ALA1027323 | B | Inhibition of human histone acetyltransferase GCN5 in U937 cell nuclear extracts assessed as remaining enzyme activity at 50 uM | Homo sapiens | 10 | ALA1136851 | cell-based format | Scientific Literature | |
| 5. | ALA1015489 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.8 mM by Western blot analysis | Homo sapiens | 1 | ALA1139367 | single protein format | Scientific Literature | |
| 6. | ALA1015490 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.2 mM by Western blot analysis | Homo sapiens | 1 | ALA1139367 | single protein format | Scientific Literature | |
| 7. | ALA1016346 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.8 mM by Western blot analysis in presence of 100 ng histone H3 | Homo sapiens | 1 | ALA1139367 | single protein format | Scientific Literature | |
| 8. | ALA1016347 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.8 mM by Western blot analysis in presence of 200 ng histone H3 | Homo sapiens | 1 | ALA1139367 | single protein format | Scientific Literature | |
| 9. | ALA1016348 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.8 mM by Western blot analysis in presence of increased concentration of acetyl-CoA | Homo sapiens | 1 | ALA1139367 | single protein format | Scientific Literature | |
| 10. | ALA1016349 | B | Inhibition of human recombinant Gcn5 assessed as reduction in acetylated histone H3 level at 0.2 mM by Western blot analysis in presence of histone H3 | Homo sapiens | 1 | ALA1139367 | single protein format | Scientific Literature | |
| 11. | ALA1738606 | F | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of GCN5L2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504398] | Homo sapiens | 13,828 | ALA1201862 | assay format | PubChem BioAssays | |
| 12. | ALA1794507 | F | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of GCN5L2: Hit confirmation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504398] | 145 | ALA1201862 | assay format | PubChem BioAssays | ||
| 13. | ALA3118017 | B | Inhibition of human recombinant histone acetyltransferase GCN5 assessed as acetylation of histone H3 at 0.15 to 0.6 mM | Homo sapiens | 1 | ALA3112473 | single protein format | Scientific Literature | |
| 14. | ALA3223010 | B | Inhibition of KAT2A (362 to 837) (unknown origin) using biotinylated histone H3 as substrate after 10 mins by TR-FRET analysis relative to control | Homo sapiens | 7 | ALA3217510 | single protein format | Scientific Literature | |
| 15. | ALA3223011 | B | Inhibition of KAT2A (362 to 837) (unknown origin) using biotinylated histone H3 as substrate at 50 uM after 10 mins by TR-FRET analysis relative to control | Homo sapiens | 1 | ALA3217510 | single protein format | Scientific Literature | |
| 16. | ALA3391520 | B | Inhibition of human GCN5 | Homo sapiens | 1 | ALA3390834 | single protein format | Scientific Literature | |
| 17. | ALA3383425 | B | Inhibition of human GCN5 by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
| 18. | ALA3424831 | B | Inhibition of recombinant GCN5 (unknown origin) | Homo sapiens | 1 | ALA3421539 | single protein format | Scientific Literature | |
| 19. | ALA3591397 | B | Binding affinity to KAT2A in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assay | Homo sapiens | 3 | ALA3588744 | cell-based format | Scientific Literature | |
| 20. | ALA3626890 | B | Inhibition of recombinant human KAT2A using biotinylated histone H3 (1 to 21 amino acid residues) as substrate at 50 uM preincubated for 10 mins followed by acetyl-CoA addition measured after 10 mins by time resolved fluorescence assay | Homo sapiens | 28 | ALA3621044 | single protein format | Scientific Literature |
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