# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA888741 | B | Inhibition of lysine methyltransferase SET7/9 at 50 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
2. | ALA1804746 | B | Inhibition of SET7-mediated methylation of histone H3 after 90 mins by scintillation counting in presence of S-adenosyl-l-[methyl-3H]methionine | 10 | single protein format | Scientific Literature | |||
3. | ALA1804754 | B | Inhibition of SET7-mediated methylation of histone H3 at 100 uM after 90 mins by scintillation counting in presence of S-adenosyl-l-[methyl-3H]methionine | 3 | single protein format | Scientific Literature | |||
4. | ALA1832595 | B | Inhibition of SETD7 assessed as hydrolysis of S-adenosyl-L-homocysteine after 2 mins by SAHH-coupled fluorescence assay | 1 | single protein format | Scientific Literature | |||
5. | ALA1953574 | B | Inhibition of HMT-set7/9 using S-adenosylmethionine and biotinylated H3 peptide at 100 uM after 1 hr | 7 | single protein format | Scientific Literature | |||
6. | ALA1799395 | B | Inhibition of methyl transferase activity of SET7/9 using biotinylated histone H3(1-21) substrate by In-vitro time resolved fluorescence immunosorbent methyltransferase assay | 1 | single protein format | Scientific Literature | |||
7. | ALA1799396 | B | Inhibition of methyl transferase activity of SET7/9 at 50 uM using biotinylated histone H3(1-21) substrate by In-vitro time resolved fluorescence immunosorbent methyltransferase assay | 6 | single protein format | Scientific Literature | |||
8. | ALA925759 | B | Inhibition of human recombinant SET7 assessed as histone H3 protein methylation at 100 uM | Homo sapiens | 24 | single protein format | Scientific Literature | ||
9. | ALA1023893 | B | Inhibition of Set7/9 lysine methyltransferase | 1 | single protein format | Scientific Literature | |||
10. | ALA1102475 | B | Inhibition of N-terminal His-tagged human recombinant SET7/9 expressed in Escherichia coli by microbeta counting | Homo sapiens | 1 | assay format | Scientific Literature | ||
11. | ALA1115314 | B | Inhibition of GST-fused human recombinant SET7 at 100 uM after 90 mins by SDS-PAGE based scintillation counting | Homo sapiens | 6 | single protein format | Scientific Literature | ||
12. | ALA1116159 | B | Inhibition of GST-fused human recombinant SET7 after 90 mins by SDS-PAGE based scintillation counting | Homo sapiens | 1 | single protein format | Scientific Literature | ||
13. | ALA1217460 | B | Activity at methyl transferase activity SET7/9 by enzyme coupled S-adenocylehomocystein detection assay | 3 | single protein format | Scientific Literature | |||
14. | ALA1292370 | B | Inhibition of human recombinant SET7/9 in cell free system assessed as monomethylation of histone H3 Lys4 residue after 1 hr in presence of 2 uM AdoMet | Homo sapiens | 5 | single protein format | Scientific Literature | ||
15. | ALA2182454 | B | Inhibition of recombinant SET7 using histone H3 as substrate at 50 uM and [3H]-SAM after 90 mins by scintillation counting | 2 | single protein format | Scientific Literature | |||
16. | ALA2209106 | B | Inhibition of SET7 using histone H3 as substrate preincubated for 10 mins followed by addition of [3H]SAM and incubated for 60 mins | 3 | single protein format | Scientific Literature | |||
17. | ALA2330203 | B | Inhibition of SETD7 (unknown origin) using histone H3 (1 to 25) as substrate after 0.5 hrs by scintillation proximity assay in presence of [3H]-S-adenosylmethionine | Homo sapiens | 1 | single protein format | Scientific Literature | ||
18. | ALA2350648 | B | Inhibition of SETD7 (unknown origin) using [3H]SAM assessed as inhibition of biotinylated-H3 (1 to 25 amino acid residues) methylation at 0.1 to 100 uM after 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
19. | ALA2434706 | B | Inhibition of human SET7/9 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
20. | ALA2434710 | B | Inhibition of human SET7/9 at 20 uM relative to control | Homo sapiens | 10 | single protein format | Scientific Literature |