| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA992488 | B | Inhibition of PCTK3 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 2. | ALA1062782 | B | Binding constant for full-length PCTK3 | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 3. | ALA1057577 | B | Inhibition of PCTK3 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 4. | ALA1102998 | B | Inhibition of PCTK3 | 1 | ALA1154951 | single protein format | Scientific Literature | ||
| 5. | ALA1166611 | B | Inhibition of PCTK3 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
| 6. | ALA1175187 | B | Inhibition of PCTK3 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 7. | ALA1244557 | B | Binding affinity to PCTK3 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 8. | ALA1827577 | B | Activity of PCTK3 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 9. | ALA1908571 | B | Binding constant for PCTK3 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 10. | ALA2215411 | B | Inhibition of PCTK3 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
| 11. | ALA2429141 | B | Competitive binding affinity to PCTK3 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | ALA2424622 | single protein format | Scientific Literature | |
| 12. | ALA3111954 | B | Inhibition of PCTK3 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
| 13. | ALA3271250 | B | Inhibition of PCTK3 (unknown origin) at 1 uM relative to control | Homo sapiens | 3 | ALA3259739 | single protein format | Scientific Literature | |
| 14. | ALA3624244 | B | Inhibition of PCTK3 (unknown origin) at 10 uM | Homo sapiens | 1 | ALA3621108 | single protein format | Scientific Literature | |
| 15. | ALA3631905 | B | Inhibition of PCTK3 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
| 16. | ALA3804612 | B | Inhibition of full length wild type human PCTK3 expressed in bacterial system assessed as enzyme activity at 1 uM relative to control | Homo sapiens | 1 | ALA3797029 | assay format | Scientific Literature | |
| 17. | ALA3991656 | B | Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry. | Homo sapiens | 27 | ALA3991601 | subcellular format | Kuster lab chemical proteomics drug profiling | |
| 18. | ALA4025294 | B | Inhibition of wild-type human full length PCTK3 (M3 to F474 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
| 19. | ALA4034447 | B | Inhibition of PCTAIRE3 Lysine 2 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
| 20. | ALA4034449 | B | Inhibition of PCTAIRE3 Lysine 1 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature |
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