# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA957098 | B | Inhibition of Mer | 1 | ALA1140952 | single protein format | Scientific Literature | ||
2. | ALA963584 | B | Binding affinity to MERTK at 10 uM by Ambit binding assay relative to control | 1 | ALA1140952 | single protein format | Scientific Literature | ||
3. | ALA964441 | B | Binding affinity to Mer at 10 uM by Ambit binding assay relative to control | 1 | ALA1140952 | single protein format | Scientific Literature | ||
4. | ALA987189 | B | Inhibition of MERTK at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
5. | ALA1025766 | B | Binding affinity to human MER at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
6. | ALA1009901 | B | Inhibition of Mer | 1 | ALA1139387 | single protein format | Scientific Literature | ||
7. | ALA1053888 | B | Inhibition of Mer assessed as residual activity at 20 uM | 1 | ALA1152913 | single protein format | Scientific Literature | ||
8. | ALA1037553 | B | Binding constant for MERTK kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
9. | ALA1047449 | B | Inhibition of MERTK assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
10. | ALA1041381 | B | Inhibition of MER at 1 uM | 1 | ALA1154622 | single protein format | Scientific Literature | ||
11. | ALA1040687 | B | Residual activity of MERTK at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
12. | ALA1041145 | B | Residual activity of MERTK at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
13. | ALA1050298 | B | Residual activity of MERTK at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
14. | ALA1100965 | B | Inhibition of MERTK at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
15. | ALA1111259 | B | Inhibition of MER at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
16. | ALA1166565 | B | Inhibition of MERTK at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
17. | ALA1174911 | B | Inhibition of MERTK at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
18. | ALA1219794 | B | Inhibition of MERTK at 1 uM by radiometric method | 2 | ALA1212904 | single protein format | Scientific Literature | ||
19. | ALA1244219 | B | Inhibition of MERTK at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
20. | ALA1244511 | B | Binding affinity to MERTK | 7 | ALA1240346 | single protein format | Scientific Literature |