# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3630491 | Binding | Inhibition of ERK5 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
2. | ALA3736806 | Binding | Inhibition of human recombinant ERK5 by LANCE assay | Homo sapiens | 1 | ALA3734740 | single protein format | Scientific Literature | |
3. | ALA3748181 | Binding | Inhibition of human ERK5 using MBP as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
4. | ALA1101124 | Binding | Inhibition of ERK5 | 1 | ALA1154951 | single protein format | Scientific Literature | ||
5. | ALA1114880 | Binding | Inhibition of ERK5 at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
6. | ALA1169225 | Binding | Inhibition of ERK5 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
7. | ALA1174415 | Binding | Inhibition of ERK5 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
8. | ALA1244832 | Binding | Binding affinity to ERK5 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
9. | ALA1827267 | Binding | Activity of ERK5 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
10. | ALA4352367 | Binding | Inhibition of human ERK5 at 10 uM using MBP as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 1 | ALA4350963 | single protein format | Scientific Literature | |
11. | ALA4357880 | Binding | Binding affinity to wild-type human partial length ERK5 (M1 to A409 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4354843 | assay format | Scientific Literature | |
12. | ALA1908585 | Binding | Binding constant for ERK5 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
13. | ALA3367929 | Binding | Inhibition of human Erk5 by Off-chip mobility shift assay | Homo sapiens | 1 | ALA3351450 | single protein format | Scientific Literature | |
14. | ALA3379503 | Binding | Inhibition of ERK5 (unknown origin) assessed as remaining enzyme activity at 10 uM by radioactive [33P]-ATP filter binding assay | Homo sapiens | 1 | ALA3351385 | single protein format | Scientific Literature | |
15. | ALA1944426 | Binding | Inhibition of human Erk5 in HL-60 cells lysate assessed as reduction of labeling of acyl-phosphate ATP probe at 100 nM | Homo sapiens | 4 | ALA1938230 | cell-based format | Scientific Literature | |
16. | ALA1670769 | Binding | Inhibition of human recombinant ERK5 in cell free system after 90 mins | Homo sapiens | 1 | ALA1667852 | single protein format | Scientific Literature | |
17. | ALA1679280 | Binding | Binding affinity to ERK5 at 10 uM by immobilized ligand displacement assay | 2 | ALA1671850 | single protein format | Scientific Literature | ||
18. | ALA1679295 | Binding | Binding affinity to ERK5 by immobilized ligand displacement assay | 1 | ALA1671850 | single protein format | Scientific Literature | ||
19. | ALA1679301 | Binding | Inhibition of EGF-induced BMK1 autophosphorylation in human HeLa cells at 0.5 uM by SDS-PAGE analysis relative to control | Homo sapiens | 19 | ALA1671850 | cell-based format | Scientific Literature | |
20. | ALA1679302 | Binding | Inhibition of EGF-induced BMK1 autophosphorylation in human HeLa cells by SDS-PAGE analysis | Homo sapiens | 19 | ALA1671850 | cell-based format | Scientific Literature |