# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3599535 | Binding | Inhibition of rat Dyrk1A using Woodtide as substrate after 40 mins by P81 membrane assay in presence of [33P]-g-ATP | Rattus norvegicus | 1 | ALA3596148 | assay format | Scientific Literature | |
2. | ALA3803248 | Binding | Inhibition of recombinant rat N-terminal GST-tagged DYRK1A (1 to 499 residues) expressed in Escherichia coli using KKISGRLSPIMTEQ-NH2 as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Rattus norvegicus | 4 | ALA3797082 | assay format | Scientific Literature | |
3. | ALA3825019 | Binding | Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using myelin basic protein as substrate incubated for 30 mins in presence of [gamma-33 ATP] by liquid scintillation counting analysis | Rattus norvegicus | 3 | ALA3822430 | assay format | Scientific Literature | |
4. | ALA1786940 | Binding | Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli assessed as assessed as incorporation of [gamma-33P]-ATP into myelin basic protein after 30 mins by scintillation counting | Rattus norvegicus | 5 | ALA1781921 | assay format | Scientific Literature | |
5. | ALA1794557 | Binding | PUBCHEM_BIOASSAY: MLPCN Dyrk1A Kinase Measured in Biochemical System Using Plate Reader - 2124-01_Inhibitor_Dose_CherryPick_Activity. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504442] | Homo sapiens | 854 | ALA1201862 | biochemical format | PubChem BioAssays | |
6. | ALA1805099 | Binding | Inhibition of rat recombinant GST-tagged DYRK1A using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation counting | Rattus norvegicus | 39 | ALA1800025 | single protein format | Scientific Literature | |
7. | ALA1805107 | Binding | Inhibition of rat recombinant GST-tagged DYRK1A using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP at 10 uM after 30 mins by scintillation counting | Rattus norvegicus | 3 | ALA1800025 | single protein format | Scientific Literature | |
8. | ALA1804241 | Binding | Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation counting | Rattus norvegicus | 36 | ALA1799982 | single protein format | Scientific Literature | |
9. | ALA1912879 | Binding | Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using myelin protein and [33P-gamma]-ATP after 30 mins by scintillation counting | Rattus norvegicus | 14 | ALA1909497 | assay format | Scientific Literature | |
10. | ALA3412950 | Binding | Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counting analysis in presence of [gamma-33P]ATP | Rattus norvegicus | 18 | ALA3407423 | assay format | Scientific Literature | |
11. | ALA1949177 | Binding | Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using myelin basic protein as substrate and [gamma-33P]ATP after 30 mins by scintillation counting | Rattus norvegicus | 20 | ALA1944600 | assay format | Scientific Literature | |
12. | ALA1044716 | Binding | Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli assessed as [gamma-33P]ATP incorporation after 10 mins by scintillation counting | Rattus norvegicus | 16 | ALA1152528 | assay format | Scientific Literature | |
13. | ALA947132 | Binding | Inhibition of rat recombinant GST-DYRK1A expressed in Escherichia coli | Rattus norvegicus | 15 | ALA1141564 | assay format | Scientific Literature | |
14. | ALA1052339 | Binding | Inhibition of rat recombinant DYRK1A expressed in Escherichia coli | Rattus norvegicus | 14 | ALA1152953 | assay format | Scientific Literature | |
15. | ALA1034401 | Binding | Inhibition of rat GST-fused Dyrk1a expressed in Escherichia coli assessed as residual enzyme activity at 10 uM | Rattus norvegicus | 9 | ALA1158396 | assay format | Scientific Literature | |
16. | ALA950841 | Binding | Inhibition of rat DYRK1a at 10 uM | Rattus norvegicus | 1 | ALA1137681 | single protein format | Scientific Literature | |
17. | ALA2032667 | Binding | Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate | Rattus norvegicus | 14 | ALA2029219 | assay format | Scientific Literature | |
18. | ALA2045871 | Binding | Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillation counting | Rattus norvegicus | 10 | ALA2040806 | assay format | Scientific Literature | |
19. | ALA2090595 | Binding | Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrate | Rattus norvegicus | 23 | ALA2086312 | assay format | Scientific Literature | |
20. | ALA2154878 | Binding | Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using [gamma-32P] ATP after 30 mins by scintillation counting | Rattus norvegicus | 8 | ALA2150858 | assay format | Scientific Literature |