# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA946634 | Binding | Inhibition of rhodopsin kinase | 1 | ALA1156449 | single protein format | Scientific Literature | ||
2. | ALA1106955 | Binding | Inhibition of GRK1-mediated bovine tubulin phosphorylation by scintillation counting | 1 | ALA1154923 | single protein format | Scientific Literature | ||
3. | ALA1169249 | Binding | Inhibition of GRK1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
4. | ALA1174440 | Binding | Inhibition of GRK1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
5. | ALA1244856 | Binding | Binding affinity to GRK1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
6. | ALA1828236 | Binding | Activity of GRK1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
7. | ALA1908595 | Binding | Binding constant for GRK1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
8. | ALA4389259 | Binding | Inhibition of wild-type human full length GRK1 (M1 to S563 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
9. | ALA4389736 | Binding | Inhibition of wild-type human full length GRK1 (M1 to S563 residues) expressed in mammalian expression system at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
10. | ALA4382540 | Binding | Binding affinity to wild-type human full length GRK1 (M1 to S563 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4382192 | assay format | Scientific Literature | |
11. | ALA3270876 | Binding | Inhibition of GRK1 (unknown origin) at 1 uM relative to control | Homo sapiens | 3 | ALA3259739 | single protein format | Scientific Literature | |
12. | ALA4365750 | Binding | Inhibition of wild-type human full length GRK1 (M1 to S563 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature | |
13. | ALA4366415 | Binding | Inhibition of human GRK1 at 100 nM using casein as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4364276 | single protein format | Scientific Literature | |
14. | ALA4377872 | Binding | Inhibition of recombinant full-length human GRK1 at 1 uM using KKKKERLLDDRHDSGLDSMKDEE as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method relative to control | Homo sapiens | 1 | ALA4376814 | single protein format | Scientific Literature | |
15. | ALA4378848 | Binding | Inhibition of full length recombinant human GRK1 at 10 uM using KKKKERLLDDRHDSGLDSMKDEE as substrate after 40 mins in presence of [gamma33P]ATP by scintillation counting method relative to control | Homo sapiens | 1 | ALA4376829 | single protein format | Scientific Literature | |
16. | ALA4379340 | Binding | Inhibition of recombinant full length human GRK1 using KKKKERLLDDRHD as substrate after 40 mins in presence of [gamma-33ATP] by radiometric scintillation counting analysis | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
17. | ALA2213533 | Binding | Inhibition of GRK1 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
18. | ALA3626279 | Binding | Inhibition of GRK1 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3621137 | single protein format | Scientific Literature | |
19. | ALA3630509 | Binding | Inhibition of GRK1 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
20. | ALA3748199 | Binding | Inhibition of human GRK1 using casein as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature |