# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1034103 | B | Inhibition of DMPK2 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
2. | ALA1060242 | B | Binding constant for DMPK2 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
3. | ALA1055294 | B | Inhibition of DMPK2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
4. | ALA1168857 | B | Inhibition of DMPK2 at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
5. | ALA1174319 | B | Inhibition of DMPK2 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
6. | ALA1244795 | B | Binding affinity to DMPK2 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
7. | ALA1827246 | B | Activity of DMPK2 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
8. | ALA1908804 | B | Binding constant for DMPK2 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
9. | ALA2216438 | B | Inhibition of DMPK2 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
10. | ALA2428157 | B | Competitive binding affinity to DMPK2 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | ALA2424622 | single protein format | Scientific Literature | |
11. | ALA3630349 | B | Inhibition of DMPK2 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
12. | ALA3749007 | B | Inhibition of human DMPK2 using [KKRPQRRYSNVF] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
13. | ALA3991648 | B | Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry. | Homo sapiens | 218 | ALA3991601 | subcellular format | Kuster lab chemical proteomics drug profiling | |
14. | ALA4025094 | B | Inhibition of wild-type human partial length DMPK2 (S46 to S408 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
15. | ALA4043905 | B | Inhibition of wild-type human partial length DMPK2 (S46 to S408 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | assay format | Scientific Literature | |
16. | ALA4054921 | B | Inhibition of wild-type human partial length DMPK2 (S46 to S408 residues) expressed in bacterial expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
17. | ALA4156984 | B | Binding affinity to wild-type human partial length DMPK2 (S46 to S408 residues) expressed in bacterial expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
18. | ALA4185763 | B | Binding affinity to wild-type human partial length DMPK2 (S46 to S408 residues) expressed in Escherichia coli BL21 at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | assay format | Scientific Literature | |
19. | ALA4230663 | B | Binding affinity to wild-type human partial length DMPK2 (S46 to S408 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
20. | ALA4264252 | B | Binding affinity to wild-type human partial length DMPK2 (S46 to S408 residues) expressed in bacterial expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4261600 | assay format | Scientific Literature |