| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA922002 | B | Activity of human MRCKbeta kinase at 1 uM | Homo sapiens | 1 | ALA1147076 | single protein format | Scientific Literature | |
| 2. | ALA992489 | B | Inhibition of MRCKB at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 3. | ALA1057486 | B | Inhibition of MRCKbeta at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
| 4. | ALA1051290 | B | Binding constant for MRCKB kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 5. | ALA1048281 | B | Inhibition of MRCKB assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 6. | ALA1066626 | B | Residual activity of CDC42BPB at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 7. | ALA1050412 | B | Residual activity of CDC42BPB at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 8. | ALA1047825 | B | Residual activity of CDC42BPB at 10 uM by microplate scintillation counting | 3 | ALA1152560 | assay format | Scientific Literature | ||
| 9. | ALA1102616 | B | Inhibition of MRCKbeta at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
| 10. | ALA1116722 | B | Inhibition of MRCKbeta at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
| 11. | ALA1166577 | B | Inhibition of MRCKB at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
| 12. | ALA1174924 | B | Inhibition of MRCKB at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 13. | ALA1219262 | B | Inhibition of MRCKbeta at 3 uM | 1 | ALA1212924 | single protein format | Scientific Literature | ||
| 14. | ALA1244388 | B | Inhibition of MRCKbeta at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 5 | ALA1240340 | single protein format | Scientific Literature | ||
| 15. | ALA1244523 | B | Binding affinity to MRCKB | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 16. | ALA1251727 | B | Inhibition of CDC42 binding protein beta at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature | ||
| 17. | ALA1259720 | B | Inhibition of MRCKbeta at 1 uM | 1 | ALA1255571 | single protein format | Scientific Literature | ||
| 18. | ALA1292330 | B | Inhibition of CDC42 BpB | 1 | ALA1287686 | single protein format | Scientific Literature | ||
| 19. | ALA1646204 | B | Inhibition of human MRCKbeta at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | ALA1641539 | single protein format | Scientific Literature | |
| 20. | ALA1826623 | B | Activity of MRCKB kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature |
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