# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1063710 | Binding | Binding constant for ERK3 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
2. | ALA1053721 | Binding | Inhibition of ERK3 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
3. | ALA1034133 | Binding | Inhibition of ERK3 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
4. | ALA1004485 | Binding | Binding affinity to human recombinant MAPK6 expressed in Escherichia coli assessed as thermal shift by differential scanning fluorimetry | Homo sapiens | 7 | ALA1140872 | assay format | Scientific Literature | |
5. | ALA1101131 | Binding | Inhibition of ERK3 | 1 | ALA1154951 | single protein format | Scientific Literature | ||
6. | ALA1169223 | Binding | Inhibition of ERK3 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
7. | ALA1174413 | Binding | Inhibition of ERK3 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
8. | ALA1244830 | Binding | Binding affinity to ERK3 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
9. | ALA1826903 | Binding | Activity of ERK3 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
10. | ALA1908584 | Binding | Binding constant for ERK3 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
11. | ALA4389228 | Binding | Inhibition of wild-type human partial length ERK3 (M1 to P413 residues) expressed in bacterial expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
12. | ALA4389705 | Binding | Inhibition of wild-type human partial length ERK3 (M1 to P413 residues) expressed in bacterial expression system at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
13. | ALA4382509 | Binding | Binding affinity to wild-type human partial length ERK3 (M1 to P413 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4382192 | assay format | Scientific Literature | |
14. | ALA4365722 | Binding | Inhibition of wild-type human partial length ERK3 (M1 to P413 residues) expressed in bacterial expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature | |
15. | ALA4375343 | Binding | Binding affinity to wild-type human partial length ERK3 (M1 to P413 residues) expressed in bacterial expression system measured after 1 hr by kinomescan method | Homo sapiens | 1 | ALA4373706 | assay format | Scientific Literature | |
16. | ALA2213998 | Binding | Inhibition of ERK3 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
17. | ALA2427151 | Binding | Competitive binding affinity to ERK3 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 4 | ALA2424622 | single protein format | Scientific Literature | |
18. | ALA2429316 | Binding | Binding affinity to ERK3 (unknown origin) | Homo sapiens | 1 | ALA2424622 | single protein format | Scientific Literature | |
19. | ALA3112109 | Binding | Inhibition of ERK3 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
20. | ALA3430817 | Binding | Delta TM value showing the stabilisation of ERK3 produced by compound binding | Homo sapiens | 156 | ALA1145498 | single protein format | Scientific Literature |