| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1826903 | B | Activity of ERK3 kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
| 2. | ALA1908584 | B | Binding constant for ERK3 kinase domain | 72 | single protein format | Scientific Literature | |||
| 3. | ALA1004485 | B | Binding affinity to human recombinant MAPK6 expressed in Escherichia coli assessed as thermal shift by differential scanning fluorimetry | Homo sapiens | 7 | assay format | Scientific Literature | ||
| 4. | ALA1034133 | B | Inhibition of ERK3 at 3 uM | 1 | single protein format | Scientific Literature | |||
| 5. | ALA1063710 | B | Binding constant for ERK3 kinase domain | Homo sapiens | 38 | single protein format | Scientific Literature | ||
| 6. | ALA1053721 | B | Inhibition of ERK3 assessed as enzyme activity at 1 uM relative to untreated control | 1 | single protein format | Scientific Literature | |||
| 7. | ALA1101131 | B | Inhibition of ERK3 | 1 | single protein format | Scientific Literature | |||
| 8. | ALA1169223 | B | Inhibition of ERK3 at 1 uM | 6 | single protein format | Scientific Literature | |||
| 9. | ALA1174413 | B | Inhibition of ERK3 at 10 uM | 2 | single protein format | Scientific Literature | |||
| 10. | ALA1244830 | B | Binding affinity to ERK3 | 7 | single protein format | Scientific Literature | |||
| 11. | ALA2213998 | B | Inhibition of ERK3 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
| 12. | ALA2427151 | B | Competitive binding affinity to ERK3 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 13. | ALA2429316 | B | Binding affinity to ERK3 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA3112109 | B | Inhibition of ERK3 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA3430817 | B | Delta TM value showing the stabilisation of ERK3 produced by compound binding | Homo sapiens | 156 | single protein format | Scientific Literature | ||
| 16. | ALA3995009 | B | Inhibition of human ERK3 (M1 to P413 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by KINOMEscan assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4025131 | B | Inhibition of wild-type human partial length ERK3 (M1 to P413 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA4043942 | B | Inhibition of wild-type human partial length ERK3 (M1 to P413 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA4055027 | B | Inhibition of wild-type human partial length ERK3 (M1 to P413 residues) expressed in bacterial expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 20. | ALA4119006 | B | Binding affinity to MAPK6 in human NCI-H358 cells at 1 uM by mass spectrometry based pull down assay | Homo sapiens | 1 | cell-based format | Scientific Literature |
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