# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA922811 | B | Activity of human DDR2 kinase at 1 uM | Homo sapiens | 1 | ALA1147076 | single protein format | Scientific Literature | |
2. | ALA973569 | B | Inhibition of DDR2 by radiometric assay | 1 | ALA1156726 | single protein format | Scientific Literature | ||
3. | ALA973717 | B | Inhibition of human DDR2 kinase assessed as residual enzyme activity at 0.1 uM | Homo sapiens | 1 | ALA1155876 | single protein format | Scientific Literature | |
4. | ALA1034100 | B | Inhibition of DDR2 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
5. | ALA1059986 | B | Inhibition of DDR2 at 10 uM | 1 | ALA1154011 | single protein format | Scientific Literature | ||
6. | ALA1061746 | B | Inhibition of DDR2 at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
7. | ALA1060180 | B | Binding constant for DDR2 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
8. | ALA1049965 | B | Binding affinity to DDR2 assessed as percentage of kinase remaining bound to the bead at 1 uM by T7 phage display based binding assay | 1 | ALA1154183 | single protein format | Scientific Literature | ||
9. | ALA1055291 | B | Inhibition of DDR2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
10. | ALA1050685 | B | Displacement of N,N'-(2,2'-(3,3'-disulfanediylbis(2,5-dioxopyrrolidine-3,1-diyl))bis(ethane-2,1-diyl))bis(2-(3-(3-tert-butyl-5-(3-naphthalen-1-ylureido)-1H-pyrazol-1-yl)phenylamino)acetamide) from inactive form of DDR2 by enzyme fragment complementation assay | 1 | ALA1156773 | single protein format | Scientific Literature | ||
11. | ALA1049458 | B | Residual activity of DDR2 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
12. | ALA1037121 | B | Residual activity of DDR2 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
13. | ALA1044289 | B | Residual activity of DDR2 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
14. | ALA1073718 | B | Inhibition of DDR2 at 3 to 6 uM relative to control | 1 | ALA1157712 | single protein format | Scientific Literature | ||
15. | ALA1107594 | B | Inhibition of DDR2 at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
16. | ALA1168854 | B | Inhibition of DDR2 at 1 uM | 8 | ALA1165965 | single protein format | Scientific Literature | ||
17. | ALA1174316 | B | Inhibition of DDR2 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
18. | ALA1244792 | B | Binding affinity to DDR2 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
19. | ALA1251490 | B | Inhibition of autophosphorylation of DDR2 expressed in HEK293 cells by ELISA | 2 | ALA1250538 | cell-based format | Scientific Literature | ||
20. | ALA1648386 | B | Inhibition of human DDR2 at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | ALA1641539 | single protein format | Scientific Literature |