# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1826997 | B | Activity of TNNI3K kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
2. | ALA1908794 | B | Binding constant for TNNI3K kinase domain | 72 | single protein format | Scientific Literature | |||
3. | ALA995066 | B | Inhibition of TNNI3K at 3 uM | 1 | single protein format | Scientific Literature | |||
4. | ALA1061932 | B | Binding constant for full-length TNNI3K | Homo sapiens | 38 | single protein format | Scientific Literature | ||
5. | ALA1059384 | B | Inhibition of TNNI3K assessed as enzyme activity at 1 uM relative to untreated control | 1 | single protein format | Scientific Literature | |||
6. | ALA1168135 | B | Inhibition of TNNI3K at 1 uM | 10 | single protein format | Scientific Literature | |||
7. | ALA1175103 | B | Inhibition of TNNI3K at 10 uM | 2 | single protein format | Scientific Literature | |||
8. | ALA1245009 | B | Binding affinity to TNNI3K | 7 | single protein format | Scientific Literature | |||
9. | ALA2209251 | B | Inhibition of TNNI3K assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
10. | ALA2428860 | B | Competitive binding affinity to TNN13K (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
11. | ALA3111559 | B | Inhibition of TNNI3K (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
12. | ALA3615798 | B | Binding affinity to TNNI3K (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
13. | ALA3615799 | B | Displacement of 5-({[2-({[3-({4-[(5-hydroxy-2-methylphenyl)amino]-2-pyrimidinyl}amino)phenyl]carbonyl}amino)-ethyl]amino}carbonyl)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid from His6-MBP-TEV-full length human TNNI3K expressed in Baculovirus expression system after 60 mins by fluorescence polarization assay | Homo sapiens | 57 | assay format | Scientific Literature | ||
14. | ALA3616263 | B | Inhibition of human myc-tagged TNNI3K autophosphorylation overexpressed in HEKMSRII cells preincubated for 30 mins followed by pervanadate solution addition measured after 20 mins by DELFIA | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
15. | ALA3816884 | B | Displacement of 5-({[2-({[3-({4-[(5-hydroxy-2-methylphenyl)amino]-2-pyrimidinyl}amino)phenyl]carbonyl}amino)-ethyl]amino}carbonyl)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid from full length human TNNI3K expressed in baculovirus system incubated for 60 mins by fluorescence polarization assay | Homo sapiens | 30 | assay format | Scientific Literature | ||
16. | ALA3816952 | B | Inhibition of human myc-tagged TNNI3K autophosphorylation overexpressed in HEKMSR2 cells incubated for 30 mins by time resolved fluorescence assay | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
17. | ALA3861903 | B | Displacement of 5-({[2-({[3-({4-[(5-hydroxy-2-methylphenyl)amino]-2-pyrimidinyl}amino)phenyl]carbonyl}amino)-ethyl]amino}carbonyl)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid from His6-MBP-TEV-full length human TNNI3K expressed in Baculovirus expression system after 60 mins by fluorescence polarization assay | Homo sapiens | 62 | assay format | Scientific Literature | ||
18. | ALA3994951 | B | Inhibition of full length human TNNI3K (M1 to S835 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by KINOMEscan assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
19. | ALA4024626 | B | Inhibition of 5-({[2-({[3-({4-[(5-hydroxy-2-methylphenyl)amino]-2-pyrimidinyl}amino)phenyl]carbonyl}amino)-ethyl]amino}carbonyl)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid binding to human full length His/MBP-fused TNNI3K expressed in baculovirus expression system after 60 mins by fluorescence polarization assay | Homo sapiens | 45 | assay format | Scientific Literature | ||
20. | ALA4024627 | B | Inhibition of human Myc-tagged TNNI3K autophosphorylation expressed in HEKMSR2 cells after 30 mins by DELFIA | Homo sapiens | 4 | cell-based format | Scientific Literature |