# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA968037 | F | Agonist activity at mouse GPR119 transfected in Xenopus dermal melanophore assessed as dispersion of melatonin-induced pigmentation | Mus musculus | 1 | ALA1139413 | assay format | Scientific Literature | |
2. | ALA1772425 | F | Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins by HTRF assay | Mus musculus | 36 | ALA1770133 | cell-based format | Scientific Literature | |
3. | ALA1772427 | F | Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation at 10 uM after 60 mins by HTRF assay | Mus musculus | 7 | ALA1770133 | cell-based format | Scientific Literature | |
4. | ALA1781105 | F | Agonist activity at mouse GPR119 expressed in HEK293 cells assessed as stimulation of cMAP level by cell-based cAMP assay | Mus musculus | 30 | ALA1777763 | cell-based format | Scientific Literature | |
5. | ALA1781106 | F | Agonist activity at mouse GPR119 expressed in HEK293 cells assessed as maximal stimulation of cMAP level by cell-based cAMP assay relative to 21 | Mus musculus | 30 | ALA1777763 | cell-based format | Scientific Literature | |
6. | ALA2014980 | F | Agonist activity at mouse GPR119 by cAMP assay | Mus musculus | 1 | ALA2010696 | assay format | Scientific Literature | |
7. | ALA2014981 | F | Agonist activity at mouse GPR119 by cAMP assay relative to oleoylethanolamide | Mus musculus | 1 | ALA2010696 | assay format | Scientific Literature | |
8. | ALA2061693 | F | Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Mus musculus | 22 | ALA2057173 | cell-based format | Scientific Literature | |
9. | ALA2061694 | F | Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay relative to AR231453 | Mus musculus | 22 | ALA2057173 | cell-based format | Scientific Literature | |
10. | ALA2089828 | F | Agonist activity at mouse GPR119 receptor assessed as increase in cAMP level after 45 mins by HTRF assay | Mus musculus | 45 | ALA2086249 | assay format | Scientific Literature | |
11. | ALA2089829 | F | Intrinsic activity at mouse GPR119 receptor assessed as increase in cAMP level after 45 mins by HTRF assay relative to oleoylethanolamide | Mus musculus | 45 | ALA2086249 | single protein format | Scientific Literature | |
12. | ALA2382538 | F | Intrinsic activity at mouse GPR119 overexpressed in HEK293S cells assessed as change in cAMP level after 45 mins by HTRF assay relative to oleoylethanolamide | Mus musculus | 16 | ALA2380211 | cell-based format | Scientific Literature | |
13. | ALA2382540 | F | Agonist activity at mouse GPR119 overexpressed in HEK293S cells assessed as change in cAMP level after 45 mins by HTRF assay | Mus musculus | 12 | ALA2380211 | cell-based format | Scientific Literature | |
14. | ALA2382542 | B | Displacement of [3H]-N-(2-fluoro-4-methylsulfonyl-phenyl)-6-[4-(3-isopropyl-1,2,4-oxadiazol-5-yl)-1-piperidyl]-5-nitro-pyrimidin-4-amine from mouse GPR119 overexpressed in baculovirus infected Sf21 cell membranes after 120 mins by scintillation counting analysis | Mus musculus | 16 | ALA2380211 | cell-based format | Scientific Literature | |
15. | ALA3106558 | F | Agonist activity at mouse GPR119 assessed as cAMP accumulation | Mus musculus | 1 | ALA3102800 | assay format | Scientific Literature | |
16. | ALA3223495 | F | Agonist activity at mouse GPR119 transfected in HEK293 cells assessed as cAMP accumulation after 45 mins incubation by HTRF assay relative to 50 uM oleoylethanolamide | Mus musculus | 18 | ALA3217541 | cell-based format | Scientific Literature | |
17. | ALA3223496 | F | Agonist activity at mouse GPR119 transfected in HEK293 cells assessed as cAMP accumulation after 45 mins incubation by HTRF assay | Mus musculus | 18 | ALA3217541 | cell-based format | Scientific Literature | |
18. | ALA3267242 | F | Agonist activity at mouse GPR119 overexpressed in CHO cells assessed as stimulation of cAMP production by HTRF assay | Mus musculus | 5 | ALA3259676 | cell-based format | Scientific Literature | |
19. | ALA3267243 | F | Agonist activity at mouse GPR119 overexpressed in CHO cells assessed as stimulation of cAMP production by HTRF assay relative to AR231453 | Mus musculus | 5 | ALA3259676 | cell-based format | Scientific Literature | |
20. | ALA3267244 | F | Agonist activity at GPR119 in mouse GLUTag cells assessed as stimulation of GLP1 secretion by CRE-luciferase reporter gene assay | Mus musculus | 5 | ALA3259676 | cell-based format | Scientific Literature |