# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA911642 | B | Activity at human PAC1 receptor in CHO cells by measuring cAMP accumulation | Homo sapiens | 2 | ALA1138207 | cell-based format | Scientific Literature | |
2. | ALA911645 | B | Displacement of [125I]PACAP27 from human PAC1 receptor expressed in CHO cells | Homo sapiens | 2 | ALA1138207 | cell-based format | Scientific Literature | |
3. | ALA949341 | B | Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cells | 22 | ALA1143199 | cell-based format | Scientific Literature | ||
4. | ALA949343 | B | Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cells at 3 uM | 13 | ALA1143199 | cell-based format | Scientific Literature | ||
5. | ALA946362 | B | Inhibition of human PACAP at 10 uM | Homo sapiens | 1 | ALA1140203 | single protein format | Scientific Literature | |
6. | ALA937783 | B | Binding affinity to human PACAP at 10 uM relative to control | Homo sapiens | 1 | ALA1140203 | single protein format | Scientific Literature | |
7. | ALA947372 | B | Displacement of radiolabeled PACAP1-38 from human PACAP | Homo sapiens | 1 | ALA1140203 | single protein format | Scientific Literature | |
8. | ALA966957 | B | Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counter | Homo sapiens | 80 | ALA1138520 | cell-based format | Scientific Literature | |
9. | ALA966958 | F | Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assay | Homo sapiens | 67 | ALA1138520 | cell-based format | Scientific Literature | |
10. | ALA966959 | F | Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as calcium mobilization by FLIPR assay | Homo sapiens | 1 | ALA1138520 | cell-based format | Scientific Literature | |
11. | ALA966960 | F | Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assay relative to PACAP38 | Homo sapiens | 68 | ALA1138520 | cell-based format | Scientific Literature | |
12. | ALA966961 | F | Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization at 1 uM by FLIPR assay | Homo sapiens | 12 | ALA1138520 | cell-based format | Scientific Literature | |
13. | ALA966962 | F | Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization at 1 uM by FLIPR assay relative to PACAP38 | Homo sapiens | 12 | ALA1138520 | cell-based format | Scientific Literature | |
14. | ALA966963 | F | Antagonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as reduction in PACAP38-induced calcium mobilization by FLIPR assay | Homo sapiens | 4 | ALA1138520 | cell-based format | Scientific Literature | |
15. | ALA966964 | F | Antagonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as reduction in PACAP38-induced calcium mobilization at 10 uM by FLIPR assay | Homo sapiens | 1 | ALA1138520 | cell-based format | Scientific Literature | |
16. | ALA1069569 | B | Displacement of [125I]PACAP1-27 from human recombinant PAC1 receptor expressed in CHO cells at 10 uM after 120 mins by scintillation counting | Homo sapiens | 1 | ALA1159093 | cell-based format | Scientific Literature | |
17. | ALA1648771 | F | Antagonist activity at human PACAPR1 expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation | Homo sapiens | 1 | ALA1641377 | cell-based format | Scientific Literature | |
18. | ALA2091422 | B | Inhibition of PACAP receptor at 5 uM by cell based assay | 1 | ALA2086382 | cell-based format | Scientific Literature | ||
19. | ALA2212553 | B | Inhibition of human PAC1 receptor at 10 uM by CEREP assay | Homo sapiens | 1 | ALA2203234 | single protein format | Scientific Literature | |
20. | ALA2209815 | B | Displacement of [125I]PACAP1-27 from human recombinant PAC1 receptor expressed in CHO cells at 10 uM after 120 mins | Homo sapiens | 1 | ALA2203205 | cell-based format | Scientific Literature |