# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1061984 | Binding | Binding constant for TLK2 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
2. | ALA1059380 | Binding | Inhibition of TLK2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
3. | ALA993452 | Binding | Binding affinity to human TLK2 at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
4. | ALA981796 | Binding | Inhibition of TLK2 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
5. | ALA1168131 | Binding | Inhibition of TLK2 at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
6. | ALA1175099 | Binding | Inhibition of TLK2 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
7. | ALA1245005 | Binding | Binding affinity to TLK2 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
8. | ALA1775241 | Binding | Inhibition of TLK2 assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma counting | 1 | ALA1773059 | single protein format | Scientific Literature | ||
9. | ALA1827555 | Binding | Activity of TLK2 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
10. | ALA1908468 | Binding | Binding constant for TLK2 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
11. | ALA4389511 | Binding | Inhibition of wild-type human partial length TLK2 (E424 to N749 residues) expressed in bacterial expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
12. | ALA4389988 | Binding | Inhibition of wild-type human partial length TLK2 (E424 to N749 residues) expressed in bacterial expression system at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
13. | ALA4382792 | Binding | Binding affinity to wild-type human partial length TLK2 (E424 to N749 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4382192 | assay format | Scientific Literature | |
14. | ALA3371266 | Binding | Inhibition of TLK2 (unknown origin) | Homo sapiens | 5 | ALA3352169 | single protein format | Scientific Literature | |
15. | ALA1942762 | Binding | Inhibition of human TLK2 in HL-60 cells lysate assessed as reduction of labeling of acyl-phosphate ATP probe at 100 nM | Homo sapiens | 4 | ALA1938230 | cell-based format | Scientific Literature | |
16. | ALA1646670 | Binding | Inhibition of human TLK2 at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | ALA1641539 | single protein format | Scientific Literature | |
17. | ALA3240760 | Binding | Inhibition of human TLK2 assessed as enzyme activity at 1 uM relative to control | Homo sapiens | 1 | ALA3232845 | single protein format | Scientific Literature | |
18. | ALA4365998 | Binding | Inhibition of wild-type human partial length TLK2 (E424 to N749 residues) expressed in bacterial expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature | |
19. | ALA4366620 | Binding | Inhibition of human TLK2 at 100 nM using casein as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4364276 | single protein format | Scientific Literature | |
20. | ALA4377929 | Binding | Inhibition of human TLK2 (387 to end residues) at 1 uM using casein as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method relative to control | Homo sapiens | 1 | ALA4376814 | single protein format | Scientific Literature |