# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2050395 | B | Inhibition of GST-tagged CARM1 expressed in escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H3 peptide after 8 mins by scintillation counting | 1 | cell-based format | Scientific Literature | |||
2. | ALA1804363 | B | Inhibition of CARM1-mediated methylation of PABP1 at 20 uM after 90 mins by scintillation counting in presence of S-adenosyl-l-[methyl-3H]methionine | 5 | single protein format | Scientific Literature | |||
3. | ALA1804593 | B | Inhibition of CARM1-mediated methylation of PABP1 after 90 mins by scintillation counting in presence of S-adenosyl-l-[methyl-3H]methionine | 10 | single protein format | Scientific Literature | |||
4. | ALA1804747 | B | Inhibition of CARM1-mediated methylation of PABP1 at 100 uM after 90 mins by scintillation counting in presence of S-adenosyl-l-[methyl-3H]methionine | 3 | single protein format | Scientific Literature | |||
5. | ALA1804748 | B | Inhibition of CARM1-mediated methylation of CA150 at 100 uM after 90 mins by scintillation counting in presence of S-adenosyl-l-[methyl-3H]methionine | 3 | single protein format | Scientific Literature | |||
6. | ALA1804749 | B | Inhibition of CARM1-mediated methylation of SMB at 100 uM after 90 mins by scintillation counting in presence of S-adenosyl-l-[methyl-3H]methionine | 3 | single protein format | Scientific Literature | |||
7. | ALA1804750 | B | Inhibition of CARM1-mediated methylation of histone H3 at 100 uM after 90 mins by scintillation counting in presence of S-adenosyl-l-[methyl-3H]methionine | 3 | single protein format | Scientific Literature | |||
8. | ALA1804758 | B | Inhibition of CARM1 expressed in tetracycline-induced human HEK293 cells coexpressing flag-tagged PABP1 assessed as inhibition of PABP1 methylation at 1 to 5 uM by SDS-PAGE analysis | 1 | cell-based format | Scientific Literature | |||
9. | ALA1804759 | B | Inhibition of CARM1-mediated prostate specific antigen promoter activity in human LNCAP cells after 48 hrs by luciferase reporter gene assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
10. | ALA1804760 | B | Inhibition of CARM1-mediated prostate specific antigen promoter activity in human LNCAP cells at 30 uM after 48 hrs by luciferase reporter gene assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
11. | ALA925758 | B | Inhibition of human recombinant CARM1 assessed as poly(A) binding protein 1 methylation at 100 uM | Homo sapiens | 25 | single protein format | Scientific Literature | ||
12. | ALA984753 | B | Inhibition of human GST-tagged CARM1 by methylation assay | Homo sapiens | 23 | single protein format | Scientific Literature | ||
13. | ALA971420 | B | Inhibition of CARM1 assessed as blockade of histone H3 methylation | 17 | single protein format | Scientific Literature | |||
14. | ALA1037272 | B | Inhibition of human CARM1 assessed as inhibition of histone3 methylation | Homo sapiens | 13 | single protein format | Scientific Literature | ||
15. | ALA1037273 | B | Inhibition of human CARM1 assessed as inhibition of HuR methylation | Homo sapiens | 1 | single protein format | Scientific Literature | ||
16. | ALA1037274 | B | Inhibition of human CARM1 assessed as inhibition of PABP methylation | Homo sapiens | 1 | single protein format | Scientific Literature | ||
17. | ALA2173353 | B | Inhibition of human CARM1 expressed in Escherichia coli BL21 (DE3) using [3H]-SAM as substrate preincubated for 10 mins before substrate addition measured after 30 mins by scintillation counter | Homo sapiens | 2 | assay format | Scientific Literature | ||
18. | ALA2175613 | B | Inhibition of CARM1 | 6 | single protein format | Scientific Literature | |||
19. | ALA2175625 | B | Inhibition of His6x-tagged PRMT4 expressed in Escherichia coli BL21 (DE3) using Histone H3(1-31) substrate in the presence of [14C] SAM assessed as residual activity at 30 uM by liquid scintillation counting | 1 | assay format | Scientific Literature | |||
20. | ALA2182448 | B | Activation of recombinant CARM1 expressed in HEK293 cells co-expressing 3XFLAG-tagged PABP1 assessed as arginine methylation of PABP1 at 50 uM after 24 hrs | Homo sapiens | 2 | cell-based format | Scientific Literature |