| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1826701 | B | Activity of SgK085 kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
| 2. | ALA1908506 | B | Binding constant for MYLK4 kinase domain | 72 | single protein format | Scientific Literature | |||
| 3. | ALA1936979 | B | Inhibition of MYLK4 at 10 uM after 1 hr by competitive binding assay | 1 | single protein format | Scientific Literature | |||
| 4. | ALA1947282 | B | Binding affinity to SGK085 assessed as change in thermal denaturation at 10 uM by thermal stability shift assay | 17 | single protein format | Scientific Literature | |||
| 5. | ALA1679284 | B | Binding affinity to MYLK4 at 10 uM by immobilized ligand displacement assay | 1 | single protein format | Scientific Literature | |||
| 6. | ALA981770 | B | Inhibition of SgK085 at 3 uM | 1 | single protein format | Scientific Literature | |||
| 7. | ALA1051352 | B | Binding constant for SgK085 kinase domain | Homo sapiens | 38 | single protein format | Scientific Literature | ||
| 8. | ALA1052963 | B | Inhibition of SgK085 assessed as enzyme activity at 1 uM relative to untreated control | 1 | single protein format | Scientific Literature | |||
| 9. | ALA1167698 | B | Inhibition of SgK085 at 1 uM | 6 | single protein format | Scientific Literature | |||
| 10. | ALA1174934 | B | Inhibition of MYLK4 at 10 uM | 2 | single protein format | Scientific Literature | |||
| 11. | ALA1244976 | B | Binding affinity to SgK085 | 7 | single protein format | Scientific Literature | |||
| 12. | ALA2215440 | B | Inhibition of MYLK4 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
| 13. | ALA2215618 | B | Binding affinity to T7-phage-tagged SgK085 by PCR analysis | 1 | single protein format | Scientific Literature | |||
| 14. | ALA2394161 | B | Competitive binding affinity to MYLK4 (unknown origin) assessed as enzyme remaining bound to anchored active-site ligand at 10 uM relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA2428993 | B | Competitive binding affinity to SgK085 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 16. | ALA2429168 | B | Binding affinity to SgK085 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA5256602 | B | Inhibition of wild type human MYLK4 at 1 uM by DiscoverX scanMAX assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA5256616 | B | Inhibition of wild type human MYLK4 in presence of ATP by radiometric kinase assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA3812027 | B | Inhibition of human MYLK4 assessed as remaining enzyme activity at 1 uM by KINOMEscan assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA4025263 | B | Inhibition of wild-type human partial length MYLK4 (V79 to S380 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature |
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