# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA950813 | B | Inhibition of IRR at 10 uM | 1 | ALA1137681 | single protein format | Scientific Literature | ||
2. | ALA945709 | B | Inhibition of human IRR at 10 uM | 1 | ALA1137681 | single protein format | Scientific Literature | ||
3. | ALA987165 | B | Inhibition of INSRR at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
4. | ALA988920 | B | Binding affinity to human IRR | Homo sapiens | 1 | ALA1151712 | single protein format | Scientific Literature | |
5. | ALA1035903 | B | Binding affinity to human IRR at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
6. | ALA1057457 | B | Inhibition of IRR at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
7. | ALA1061175 | B | Binding constant for INSRR kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
8. | ALA1056924 | B | Inhibition of IRR assessed as remaining enzyme activity at 3 uM relative to DMSO | 1 | ALA1154183 | single protein format | Scientific Literature | ||
9. | ALA1055348 | B | Inhibition of IRR assessed as remaining enzyme activity at 1 uM relative to DMSO | 1 | ALA1154183 | single protein format | Scientific Literature | ||
10. | ALA1053754 | B | Inhibition of INSRR assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
11. | ALA1041371 | B | Inhibition of IRR at 1 uM | 1 | ALA1154622 | single protein format | Scientific Literature | ||
12. | ALA1044625 | B | Inhibition of IRR assessed as residual activity at 10 uM by Cherenkov counting relative to control in presence of 5 uM ATP | 2 | ALA1155278 | single protein format | Scientific Literature | ||
13. | ALA1050752 | B | Inhibition of IRR assessed as residual activity at 0.1 uM by Cherenkov counting relative to control in presence of 5 uM ATP | 2 | ALA1155278 | single protein format | Scientific Literature | ||
14. | ALA1040663 | B | Residual activity of INSRR at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
15. | ALA1041121 | B | Residual activity of INSRR at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
16. | ALA1046835 | B | Residual activity of INSRR at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
17. | ALA1073302 | B | Inhibition of INSR | 1 | ALA1153138 | single protein format | Scientific Literature | ||
18. | ALA1100364 | B | Inhibition of INSRR at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
19. | ALA1111197 | B | Inhibition of IRR at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
20. | ALA1104329 | B | Inhibition of IRR at 10 uM assessed as residual activity by [33P]ATP radioactive filter binding assay relative to control | 2 | ALA1156950 | single protein format | Scientific Literature |