# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1033256 | B | Inhibition of CSNK1A1L at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
2. | ALA1063703 | B | Binding constant for full-length CSNK1A1L | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
3. | ALA1052900 | B | Inhibition of CSNK1A1L assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
4. | ALA1168838 | B | Inhibition of CSNK1A1L at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
5. | ALA1174184 | B | Inhibition of CSNK1A1L at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
6. | ALA1908420 | B | Binding constant for CSNK1A1L kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
7. | ALA2209314 | B | Inhibition of CSNK1A1L assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
8. | ALA2428168 | B | Competitive binding affinity to CSNK1A1L (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 4 | ALA2424622 | single protein format | Scientific Literature | |
9. | ALA3112112 | B | Inhibition of CSNK1A1L (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
10. | ALA3386800 | B | Inhibition of CSNK1A1L (unknown origin) assessed as residual enzyme activity at 10 uM | Homo sapiens | 2 | ALA3352555 | single protein format | Scientific Literature | |
11. | ALA3424694 | B | Inhibition of human Casein kinase 1 alpha 1-like assessed as residual activity at 10 uM relative to control | Homo sapiens | 4 | ALA3421615 | single protein format | Scientific Literature | |
12. | ALA3812037 | B | Inhibition of full-length human CSNK1A1L expressed in bacterial system assessed as remaining enzyme activity at 1 uM by KINOMEscan assay | Homo sapiens | 1 | ALA3808325 | assay format | Scientific Literature | |
13. | ALA4025075 | B | Inhibition of wild-type human full length CSNK1A1L (M1 to N337 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
14. | ALA4043886 | B | Inhibition of wild-type human full length CSNK1A1L (M1 to N337 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | assay format | Scientific Literature | |
15. | ALA4156965 | B | Binding affinity to wild-type human full length CSNK1A1L (M1 to N337 residues) expressed in bacterial expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
16. | ALA4185744 | B | Binding affinity to wild-type human full length CSNK1A1L (M1 to N337 residues) expressed in Escherichia coli BL21 at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | assay format | Scientific Literature | |
17. | ALA4230644 | B | Binding affinity to wild-type human full length CSNK1A1L (M1 to N337 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
18. | ALA4264233 | B | Binding affinity to wild-type human full length CSNK1A1L (M1 to N337 residues) expressed in bacterial expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4261600 | assay format | Scientific Literature | |
19. | ALA4307748 | B | Binding affinity to wild-type human full length CSNK1A1L (M1 to N337 residues) expressed in bacterial expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4304811 | assay format | Scientific Literature | |
20. | ALA4327643 | B | Inhibition of human CK1a1L assessed as residual activity at 1 uM using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | ALA4325871 | single protein format | Scientific Literature |