# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1061080 | Binding | Binding constant for MYO3A kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
2. | ALA1048290 | Binding | Inhibition of MYO3A assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
3. | ALA987208 | Binding | Inhibition of MYO3A at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
4. | ALA1166586 | Binding | Inhibition of MYO3A at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
5. | ALA1174935 | Binding | Inhibition of MYO3A at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
6. | ALA1244532 | Binding | Binding affinity to MYO3A | 7 | ALA1240346 | single protein format | Scientific Literature | ||
7. | ALA1827250 | Binding | Activity of MYO3A kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
8. | ALA1908801 | Binding | Binding constant for MYO3A kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
9. | ALA4389361 | Binding | Inhibition of wild-type human partial length MYO3A (M1 to K338 residues) expressed in bacterial expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
10. | ALA4389838 | Binding | Inhibition of wild-type human partial length MYO3A (M1 to K338 residues) expressed in bacterial expression system at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
11. | ALA4382642 | Binding | Binding affinity to wild-type human partial length MYO3A (M1 to K338 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4382192 | assay format | Scientific Literature | |
12. | ALA4365849 | Binding | Inhibition of wild-type human partial length MYO3A (M1 to K338 residues) expressed in bacterial expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature | |
13. | ALA4366504 | Binding | Inhibition of human MYO3A at 100 nM using MBP as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4364276 | single protein format | Scientific Literature | |
14. | ALA2215439 | Binding | Inhibition of MYO3A assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
15. | ALA2429662 | Binding | Competitive binding affinity to MYO3A (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | ALA2424622 | single protein format | Scientific Literature | |
16. | ALA4025264 | Binding | Inhibition of wild-type human partial length MYO3A (M1 to K338 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
17. | ALA4034416 | Binding | Inhibition of MYO3A (unknown origin) labeling at conserved lysine2 at 10 uM relative to control | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
18. | ALA4044075 | Binding | Inhibition of wild-type human partial length MYO3A (M1 to K338 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | assay format | Scientific Literature | |
19. | ALA4055060 | Binding | Inhibition of wild-type human partial length MYO3A (M1 to K338 residues) expressed in bacterial expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
20. | ALA4157154 | Binding | Binding affinity to wild-type human partial length MYO3A (M1 to K338 residues) expressed in bacterial expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature |