# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1032252 | B | Inhibition of ANKK1 at 3 uM | 1 | single protein format | Scientific Literature | |||
2. | ALA1060235 | B | Binding constant for ANKK1 kinase domain | Homo sapiens | 38 | single protein format | Scientific Literature | ||
3. | ALA1059259 | B | Inhibition of ANKK1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | single protein format | Scientific Literature | |||
4. | ALA1168787 | B | Inhibition of ANKK1 at 1 uM | 6 | single protein format | Scientific Literature | |||
5. | ALA1174069 | B | Inhibition of ANKK1 at 10 uM | 2 | single protein format | Scientific Literature | |||
6. | ALA1244725 | B | Binding affinity to ANKK1 | 7 | single protein format | Scientific Literature | |||
7. | ALA1826893 | B | Activity of ANKK1 kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
8. | ALA1908432 | B | Binding constant for ANKK1 kinase domain | 72 | single protein format | Scientific Literature | |||
9. | ALA2176624 | B | Inhibition of ANKK1 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
10. | ALA2212075 | B | Inhibition of ANKK1 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
11. | ALA2428327 | B | Competitive binding affinity to ANKK1 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
12. | ALA3112122 | B | Inhibition of ANKK1 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
13. | ALA4025014 | B | Inhibition of wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
14. | ALA4043825 | B | Inhibition of wild-type human partial length ANKK1 (M1 to A305 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
15. | ALA4055259 | B | Inhibition of wild-type human partial length SGK288 (M1 to A305 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
16. | ALA4156904 | B | Binding affinity to wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
17. | ALA4185683 | B | Binding affinity to wild-type human partial length ANKK1 (M1 to A305 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
18. | ALA4230583 | B | Binding affinity to wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
19. | ALA4264172 | B | Binding affinity to wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
20. | ALA4307689 | B | Binding affinity to wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature |