# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1060235 | B | Binding constant for ANKK1 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
2. | ALA1059259 | B | Inhibition of ANKK1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
3. | ALA1032252 | B | Inhibition of ANKK1 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
4. | ALA1168787 | B | Inhibition of ANKK1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
5. | ALA1174069 | B | Inhibition of ANKK1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
6. | ALA1244725 | B | Binding affinity to ANKK1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
7. | ALA1826893 | B | Activity of ANKK1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
8. | ALA1908432 | B | Binding constant for ANKK1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
9. | ALA4389111 | B | Inhibition of wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
10. | ALA4389588 | B | Inhibition of wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
11. | ALA4382392 | B | Binding affinity to wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4382192 | assay format | Scientific Literature | |
12. | ALA4365607 | B | Inhibition of wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature | |
13. | ALA2176624 | B | Inhibition of ANKK1 assessed as residual activity at 10 uM relative to control | 1 | ALA2169853 | single protein format | Scientific Literature | ||
14. | ALA2212075 | B | Inhibition of ANKK1 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
15. | ALA2428327 | B | Competitive binding affinity to ANKK1 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | ALA2424622 | single protein format | Scientific Literature | |
16. | ALA3112122 | B | Inhibition of ANKK1 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
17. | ALA4025014 | B | Inhibition of wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
18. | ALA4043825 | B | Inhibition of wild-type human partial length ANKK1 (M1 to A305 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature | |
19. | ALA4055259 | B | Inhibition of wild-type human partial length SGK288 (M1 to A305 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
20. | ALA4156904 | B | Binding affinity to wild-type human partial length ANKK1 (M1 to A305 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature |