| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA997767 | Binding | Displacement of [I125]MIT from PKR2 expressed in CHO cell membrane | 3 | ALA1140216 | cell-based format | Scientific Literature | ||
| 2. | ALA998632 | Functional | Antagonist activity at PKR2 expressed in CHO cell membrane assessed as reduction of Bv8-induced increase in intracellular calcium level at 100 nM | 1 | ALA1140216 | cell-based format | Scientific Literature | ||
| 3. | ALA998634 | Functional | Antagonist activity at PKR2 expressed in CHO cell membrane assessed as reduction of Bv8-induced increase in intracellular calcium level at 300 nM | 1 | ALA1140216 | cell-based format | Scientific Literature | ||
| 4. | ALA998636 | Functional | Antagonist activity at PKR2 expressed in CHO cell membrane assessed as reduction of Bv8-induced increase in intracellular calcium level at 10 uM | 1 | ALA1140216 | cell-based format | Scientific Literature | ||
| 5. | ALA998638 | Functional | Antagonist activity at PKR2 expressed in CHO cell membrane assessed as reduction of Bv8-induced increase in intracellular calcium level at 1 mM | 1 | ALA1140216 | cell-based format | Scientific Literature | ||
| 6. | ALA998640 | Functional | Antagonist activity at PKR2 expressed in CHO cell membrane assessed as reduction of Bv8-induced increase in intracellular calcium level at 100 uM | 1 | ALA1140216 | cell-based format | Scientific Literature | ||
| 7. | ALA4883575 | Binding | PRESTO-Tango GPCRome screening (PK2) | 1 | ALA4507309 | single protein format | Donated Chemical Probes - SGC Frankfurt |
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