| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1032272 | B | Inhibition of CIT at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 2. | ALA1062838 | B | Binding constant for CIT kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 3. | ALA1052893 | B | Inhibition of CIT assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 4. | ALA1038691 | B | Inhibition of CIT | 1 | ALA1154622 | single protein format | Scientific Literature | ||
| 5. | ALA1114869 | B | Inhibition of CRIK at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
| 6. | ALA1168831 | B | Inhibition of CIT at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
| 7. | ALA1174176 | B | Inhibition of CIT at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 8. | ALA1244769 | B | Binding affinity to CIT | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 9. | ALA1826899 | B | Activity of CIT kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 10. | ALA1908762 | B | Binding constant for CIT kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 11. | ALA2014914 | B | Inhibition of CRIK at 10 uM | 1 | ALA2010722 | single protein format | Scientific Literature | ||
| 12. | ALA2209323 | B | Inhibition of CIT assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
| 13. | ALA2394172 | B | Competitive binding affinity to CIT (unknown origin) assessed as enzyme remaining bound to anchored active-site ligand at 10 uM relative to control | Homo sapiens | 1 | ALA2390846 | single protein format | Scientific Literature | |
| 14. | ALA2428169 | B | Competitive binding affinity to CIT (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 4 | ALA2424622 | single protein format | Scientific Literature | |
| 15. | ALA2429324 | B | Binding affinity to CIT (unknown origin) | Homo sapiens | 1 | ALA2424622 | single protein format | Scientific Literature | |
| 16. | ALA3112113 | B | Inhibition of CIT (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
| 17. | ALA3370292 | B | Inhibition of human CRIK by Off-chip mobility shift assay | Homo sapiens | 1 | ALA3351450 | single protein format | Scientific Literature | |
| 18. | ALA3631913 | B | Inhibition of STK21 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
| 19. | ALA3991667 | B | Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry. | Homo sapiens | 243 | ALA3991601 | subcellular format | Kuster lab chemical proteomics drug profiling | |
| 20. | ALA4025066 | B | Inhibition of wild-type human partial length CIT (M68 to E432 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature |
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