| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA927943 | B | Activity of human BrSK1 kinase at 1 uM | Homo sapiens | 1 | ALA1147076 | single protein format | Scientific Literature | |
| 2. | ALA1032266 | B | Inhibition of BRSK1 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 3. | ALA1061565 | B | Inhibition of BRSK1 at 1 uM | 2 | ALA1153487 | single protein format | Scientific Literature | ||
| 4. | ALA1060966 | B | Inhibition of BRSK1 at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
| 5. | ALA1061135 | B | Binding constant for BRSK1 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 6. | ALA1052868 | B | Inhibition of BRSK1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 7. | ALA1041337 | B | Inhibition of BRSK1 at 1 uM | 1 | ALA1154622 | single protein format | Scientific Literature | ||
| 8. | ALA1066617 | B | Residual activity of BRSK1 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 9. | ALA1050403 | B | Residual activity of BRSK1 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 10. | ALA1047816 | B | Residual activity of BRSK1 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 11. | ALA1102608 | B | Inhibition of BRSK1 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
| 12. | ALA1114028 | B | Inhibition of BRSK1 at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
| 13. | ALA1116003 | B | Inhibition of BRSK1 at 10 uM assessed as residual activity by [33P]ATP radioactive filter binding assay relative to control | 2 | ALA1156950 | single protein format | Scientific Literature | ||
| 14. | ALA1168804 | B | Inhibition of BRSK1 at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
| 15. | ALA1174086 | B | Inhibition of BRSK1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 16. | ALA1244380 | B | Inhibition of BRSK1 at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 5 | ALA1240340 | single protein format | Scientific Literature | ||
| 17. | ALA1244742 | B | Binding affinity to BRSK1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 18. | ALA1251640 | B | Inhibition of BRSK1 at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature | ||
| 19. | ALA1648524 | B | Inhibition of BRSK1 assessed as residual activity at 10 uM | 3 | ALA1641579 | single protein format | Scientific Literature | ||
| 20. | ALA1648182 | B | Inhibition of human BrSK1 at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | ALA1641539 | single protein format | Scientific Literature |
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