| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA999776 | B | Binding affinity to human CDK8 at 5 uM | Homo sapiens | 2 | ALA1136966 | single protein format | Scientific Literature | |
| 2. | ALA1032234 | B | Inhibition of CDK8 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 3. | ALA1051283 | B | Binding constant for CDK8 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 4. | ALA1052888 | B | Inhibition of CDK8 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 5. | ALA1101138 | B | Inhibition of CDK8 | 1 | ALA1154951 | single protein format | Scientific Literature | ||
| 6. | ALA1168824 | B | Inhibition of CDK8 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
| 7. | ALA1174168 | B | Inhibition of CDK8 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 8. | ALA1244762 | B | Binding affinity to CDK8 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 9. | ALA1786914 | B | Binding affinity to human CDK8 at 10 uM incubated for 1 hr by kinase binding assay relative to untreated control | Homo sapiens | 3 | ALA1782045 | single protein format | Scientific Literature | |
| 10. | ALA1787153 | B | Binding affinity to human CDK8 incubated for 1 hr by kinase binding assay | Homo sapiens | 1 | ALA1782045 | single protein format | Scientific Literature | |
| 11. | ALA1826943 | B | Activity of CDK8 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 12. | ALA1908526 | B | Binding constant for CDK8 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 13. | ALA1963824 | F | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CDK8 | 422 | ALA1201862 | assay format | PubChem BioAssays | ||
| 14. | ALA2209330 | B | Inhibition of CDK8 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
| 15. | ALA2422448 | B | Inhibition of CDK8 in human PC3 cell lysates at 10 uM using desthiobiotin-tagged ATP probe AX9989 followed by trypsinization by LC/MS analysis | Homo sapiens | 12 | ALA2417377 | single protein format | Scientific Literature | |
| 16. | ALA2428173 | B | Competitive binding affinity to CDK8 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | ALA2424622 | single protein format | Scientific Literature | |
| 17. | ALA3101306 | B | Inhibition of active state of CDK8 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3098110 | single protein format | Scientific Literature | |
| 18. | ALA3112117 | B | Inhibition of CDK8 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
| 19. | ALA3268854 | B | Inhibition of CDK8 (unknown origin) at 1 uM relative to control | Homo sapiens | 3 | ALA3259739 | single protein format | Scientific Literature | |
| 20. | ALA3387826 | B | Inhibition of CDK8 (unknown origin) | Homo sapiens | 4 | ALA3352406 | single protein format | Scientific Literature |
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