# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA940040 | B | Inhibition of human MRP2 expressed in MDCK2 cells assessed as increase in intracellular CMF fluorescence by CMFDA assay | Homo sapiens | 7 | ALA1147049 | cell-based format | Scientific Literature | |
2. | ALA940043 | B | Inhibition of human MRP2 expressed in MDCK2 cells assessed as increase in intracellular CMF fluorescence at 10 uM by CMFDA assay | Homo sapiens | 6 | ALA1147049 | cell-based format | Scientific Literature | |
3. | ALA940046 | B | Inhibition of human MRP2 expressed in MDCK2 cells assessed as increase in intracellular CMF fluorescence at 16.7 uM by CMFDA assay | Homo sapiens | 1 | ALA1147049 | cell-based format | Scientific Literature | |
4. | ALA975399 | B | Inhibition of human MRP2 expressed in dog MDCK2 cells | Homo sapiens | 8 | ALA1140042 | cell-based format | Scientific Literature | |
5. | ALA957853 | B | Inhibition of ABCC2 overexpressed in MDCK cells at 100 uM by flow cytometric-based chloromethylfluorescein-diacetate accumulation assay | 10 | ALA1140935 | cell-based format | Scientific Literature | ||
6. | ALA957854 | B | Inhibition of ABCC2 overexpressed in MDCK cells at 100 uM up to 50 uM by flow cytometric-based chloromethylfluorescein-diacetate accumulation assay | 7 | ALA1140935 | cell-based format | Scientific Literature | ||
7. | ALA1006005 | B | Effect on human MRP2-mediated estradiol-17-beta-glucuronide transport in Sf9 cells inverted membrane vesicles relative to control | Homo sapiens | 189 | ALA1150338 | cell-based format | Scientific Literature | |
8. | ALA1006006 | B | Inhibition of human MRP2-mediated estradiol-17-beta-glucuronide transport in Sf9 cells inverted membrane vesicles | Homo sapiens | 1 | ALA1150338 | cell-based format | Scientific Literature | |
9. | ALA1062296 | B | Inhibition of MRP2 | 3 | ALA1152445 | single protein format | Scientific Literature | ||
10. | ALA1177213 | B | Inhibition of MRP2 expressed in human A2780 cells at 10 uM relative to control | 16 | ALA1177685 | cell-based format | Scientific Literature | ||
11. | ALA1692698 | B | Inhibition of MRP2 expressed in MDCK2 cells assessed as cell growth inhibition by calcein and pheophorbide A efflux assays | 1 | ALA1687850 | cell-based format | Scientific Literature | ||
12. | ALA1692720 | B | Activity at MRP2 | 4 | ALA1687850 | single protein format | Scientific Literature | ||
13. | ALA1743160 | A | Substrates of transporters of clinical importance in the absorption and disposition of drugs, MRP2 | Homo sapiens | 6 | ALA1743141 | single protein format | Scientific Literature | |
14. | ALA1743179 | A | Inhibitors of transporters of clinical importance in the absorption and disposition of drugs, MRP2 | Homo sapiens | 4 | ALA1743141 | single protein format | Scientific Literature | |
15. | ALA1953008 | B | Binding affinity to MRP2 expressed in MDCK2 cells coexpressing OATP1B1 | 1 | ALA1949499 | cell-based format | Scientific Literature | ||
16. | ALA1953009 | B | Binding affinity to MRP2 expressed in MDCK2 cells coexpressing OATP1B3 | 1 | ALA1949499 | cell-based format | Scientific Literature | ||
17. | ALA2013263 | A | Inhibition of MRP2 | 1 | ALA2010675 | single protein format | Scientific Literature | ||
18. | ALA2077555 | F | TP_TRANSPORTER: secretion into apical vacuoles in Hep G2 cells | 4 | ALA2073786 | cell-based format | TP-search Transporter Database | ||
19. | ALA2077556 | F | TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicles from MRP2-expressing LLC PK1 cells | 4 | ALA2073997 | cell membrane format | TP-search Transporter Database | ||
20. | ALA2077557 | F | TP_TRANSPORTER: inhibition of EGCG in MRP2-expressing MDCKII cells | 4 | ALA2074563 | cell-based format | TP-search Transporter Database |