# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA831102 | B | Inhibition of estrogen-related receptor alpha Gal4 activity | 1 | single protein format | Scientific Literature | |||
2. | ALA827660 | B | Inhibition of estrogen-related receptor alpha Gal4 activity | 18 | single protein format | Scientific Literature | |||
3. | ALA828552 | B | Inhibition of estrogen-related receptor alpha in FP assay | 1 | single protein format | Scientific Literature | |||
4. | ALA832619 | B | Inhibition of estrogen-related receptor alpha Gal4 activity; not active | 3 | single protein format | Scientific Literature | |||
5. | ALA874762 | B | Percent inhibition of estrogen-related receptor alpha Gal4 activity at 10 uM | 18 | single protein format | Scientific Literature | |||
6. | ALA831934 | B | Percent inhibition of estrogen-related receptor alpha Gal4 activity at 10 uM; not active | 2 | single protein format | Scientific Literature | |||
7. | ALA837152 | F | Fold activation of estrogen-related receptor alpha at 3 uM in cell-based reporter gene assay | 1 | cell-based format | Scientific Literature | |||
8. | ALA837725 | F | Fold activation of estrogen-related receptor alpha at 10 uM in cell-based reporter gene assay | 1 | cell-based format | Scientific Literature | |||
9. | ALA837726 | F | Fold activation of estrogen-related receptor alpha at 30 uM in cell-based reporter gene assay | 1 | cell-based format | Scientific Literature | |||
10. | ALA826312 | F | Fold activation of estrogen-related receptor alpha at 100 nM in cell-based reporter gene assay | 1 | cell-based format | Scientific Literature | |||
11. | ALA860923 | B | Binding affinity to human ERalpha relative to estradiol by radiometric binding assay | Homo sapiens | 24 | single protein format | Scientific Literature | ||
12. | ALA888441 | B | Binding affinity to ERalpha | 1 | single protein format | Scientific Literature | |||
13. | ALA941998 | B | Displacement of [3H]estradiol from estrogen receptor alpha at 10 uM | Homo sapiens | 19 | single protein format | Scientific Literature | ||
14. | ALA1918098 | B | Agonist activity at human ERRalpha ligand binding domain expressed in human 293FT cells coexpressing Gal4 DNA binding domain assessed as increased transcriptional activity at 10 uM after 24 hrs by dual luciferase reporter gene assay relative to control | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
15. | ALA1918099 | B | Agonist activity at human ERRalpha ligand binding domain expressed in human 293FT cells coexpressing Gal4 DNA binding domain assessed as increased transcriptional activity after 24 hrs by dual luciferase reporter gene assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
16. | ALA1918209 | B | Inverse agonist activity at human ERRalpha ligand binding domain expressed in human 293FT cells coexpressing with Gal4 DNA binding domain assessed as inhibition of transcriptional activity at 10 uM after 24 hrs by dual luciferase reporter gene assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
17. | ALA1918210 | B | Agonist activity at human ERRalpha ligand binding domain expressed in human 293FT cells coexpressing with Gal4 DNA binding domain assessed as increased transcriptional activity at 1 to 5 uM after 24 hrs by dual luciferase reporter gene assay in presence of kaempferol | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
18. | ALA886438 | B | Inhibition of human ERalpha | Homo sapiens | 21 | single protein format | Scientific Literature | ||
19. | ALA902796 | B | Effect on interaction between ERRalpha ligand binding domain and RIP140 at 30 uM by FRET assay | Homo sapiens | 18 | single protein format | Scientific Literature | ||
20. | ALA902798 | B | Activity at human ERRalpha expressed in HeLa cells assessed as estrogen response element activation at 50 uM after 24 ro 30 hrs by luciferase reporter gene assay | Homo sapiens | 18 | cell-based format | Scientific Literature |