| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA895919 | B | Inhibition of E2K2 | Homo sapiens | 1 | ALA1148766 | single protein format | Scientific Literature | |
| 2. | ALA992504 | B | Inhibition of PRKR at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 3. | ALA1062867 | B | Binding constant for PRKR kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 4. | ALA1052934 | B | Inhibition of PRKR assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 5. | ALA1038365 | B | Inhibition of PKR | 1 | ALA1155349 | single protein format | Scientific Literature | ||
| 6. | ALA1049467 | B | Residual activity of EIF2AK2 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 7. | ALA1037130 | B | Residual activity of EIF2AK2 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 8. | ALA1044298 | B | Residual activity of EIF2AK2 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 9. | ALA1101127 | B | Inhibition of PRKR | 1 | ALA1154951 | single protein format | Scientific Literature | ||
| 10. | ALA1103222 | B | Inhibition of PKR at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
| 11. | ALA1166830 | B | Inhibition of PRKR at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
| 12. | ALA1175240 | B | Inhibition of PRKR at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 13. | ALA1226713 | B | Inhibition of PKR-mediated p53 phosphorylation | 1 | ALA1221185 | single protein format | Scientific Literature | ||
| 14. | ALA1244945 | B | Binding affinity to PRKR | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 15. | ALA1805140 | B | Inhibition of human recombinant PKR autophosphorylation using poly[I:C] after 10 mins by luminescent assay | Homo sapiens | 81 | ALA1799935 | single protein format | Scientific Literature | |
| 16. | ALA1805144 | B | Competitive inhibition of human recombinant PKR | Homo sapiens | 1 | ALA1799935 | single protein format | Scientific Literature | |
| 17. | ALA1827283 | B | Activity of PRKR kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 18. | ALA1838133 | B | Inhibition of human PKR in HL60 cells lysate at 10 uM using post probe-labeling by LC-MS/MS analysis relative to control | Homo sapiens | 5 | ALA1833925 | cell-based format | Scientific Literature | |
| 19. | ALA1908593 | B | Binding constant for PRKR kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 20. | ALA1942757 | B | Inhibition of human PKR in HL-60 cells lysate assessed as reduction of labeling of acyl-phosphate ATP probe at 100 nM | Homo sapiens | 4 | ALA1938230 | cell-based format | Scientific Literature |
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