| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA995026 | B | Inhibition of PFTAIRE2 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 2. | ALA1057581 | B | Inhibition of PFTAIRE2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 3. | ALA1166615 | B | Inhibition of PFTAIRE2 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
| 4. | ALA1175193 | B | Inhibition of PFTAIRE2 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 5. | ALA1244561 | B | Binding affinity to PFTAIRE2 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 6. | ALA1826682 | B | Activity of PFTAIRE2 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 7. | ALA1908415 | B | Binding constant for PFTAIRE2 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 8. | ALA2214970 | B | Inhibition of PFTAIRE2 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
| 9. | ALA4025300 | B | Inhibition of wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
| 10. | ALA4044111 | B | Inhibition of wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | assay format | Scientific Literature | |
| 11. | ALA4055234 | B | Inhibition of wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in bacterial expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
| 12. | ALA4118447 | B | Inhibition of PFTAIRE2 in human SKCO1 cells at 1 uM after 4 hrs using biotin labeled DLKPQNLLISHLGELK probe by mass-spectrometric analysis relative to control | Homo sapiens | 3 | ALA4118021 | cell-based format | Scientific Literature | |
| 13. | ALA4157190 | B | Binding affinity to wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in bacterial expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
| 14. | ALA4185969 | B | Binding affinity to wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in Escherichia coli BL21 at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | assay format | Scientific Literature | |
| 15. | ALA4230869 | B | Binding affinity to wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
| 16. | ALA4264458 | B | Binding affinity to wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in bacterial expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4261600 | assay format | Scientific Literature | |
| 17. | ALA4307968 | B | Binding affinity to wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in bacterial expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4304811 | assay format | Scientific Literature | |
| 18. | ALA4333553 | B | Binding affinity to wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4330132 | assay format | Scientific Literature | |
| 19. | ALA4358047 | B | Binding affinity to wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4354843 | assay format | Scientific Literature | |
| 20. | ALA4365885 | B | Inhibition of wild-type human full length PFTAIRE2 (M1 to W384 residues) expressed in bacterial expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature |
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