| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1930561 | F | Activation of C-terminal HA epitope tagged human TAAR1 expressed in RD-HGA16 cells co-expressing Gq protein, Galpha16 by cAMP accumulation assay | Homo sapiens | 19 | cell-based format | Scientific Literature | ||
| 2. | ALA1930651 | F | Activation of human TAAR1 expressed in CHOK1 cells co-expressing Gq protein, Galpha16 using calcium4 dye by microplate reader | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA1930658 | F | Activation of human TAAR1 expressed in Syrian hamster AV12-664 cells co-expressing GalphaS protein assessed as accumulation of cAMP after 30 mins using cAMP XS EA/CL as substrate by luminescence method in presence of RX821002 and alprenolol | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 4. | ALA1930659 | F | Activation of human TAAR1 expressed in human HEK293T cells assessed as cAMP accumulation after 10 mins by BRET assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 5. | ALA1670082 | B | Inhibition of human TAAR1 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA1670128 | F | Antagonist activity at human TAAR1 assessed as reversal of endogenous beta-PEA effect | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 7. | ALA1670255 | F | Antagonist activity at humanTAAR1 assessed as residual stimulation by in vitro cAMP functional assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA989986 | F | Agonist activity at human trace amine associated receptor 1 expressed in RD-HGA16 CHO-K1 cells coexpressed with Galpha16 protein assessed as internal calcium mobilization by calcium 3 assay | Homo sapiens | 69 | cell-based format | Scientific Literature | ||
| 9. | ALA989987 | F | Agonist activity at human trace amine associated receptor 1 expressed in RD-HGA16 CHO-K1 cells coexpressed with Galpha16 protein assessed as internal calcium mobilization by calcium 3 assay relative to 2-phenylethanamine | Homo sapiens | 68 | cell-based format | Scientific Literature | ||
| 10. | ALA989988 | F | Agonist activity at human trace amine associated receptor 1 expressed in AV12-664 cells coexpressed with rat GalphaS protein assessed as cAMP accumulation | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 11. | ALA989989 | F | Agonist activity at human trace amine associated receptor 1 expressed in AV12-664 cells coexpressed with rat Galpha16 protein assessed as cAMP accumulation relative to 2-phenylethanamine | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 12. | ALA1048859 | F | Activation of human TAAR1 expressed in CHOK1 cells assessed as cAMP accumulation at 0.1 to 1 uM | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 13. | ALA1048860 | F | Activation of human TAAR1 expressed in CHOK1 cells coexpressing Galpha16 assessed as calcium accumulation at 0.1 to 1 uM relative to beta-phenethylamine | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 14. | ALA1048862 | F | Activation of human TAAR1 expressed in CHOK1 cells assessed as cAMP accumulation at 10 uM relative to beta-phenethylamine | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 15. | ALA1048863 | F | Activation of human TAAR1 expressed in CHOK1 cells coexpressing Galpha16 assessed as calcium accumulation at 10 uM relative to beta-phenethylamine | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 16. | ALA1048864 | F | Activation of human TAAR1 expressed in CHOK1 cells coexpressing Galpha16 assessed as calcium accumulation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA1048866 | F | Activation of human TAAR1 expressed in CHOK1 cells coexpressing Galpha16 assessed as calcium accumulation relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA2213071 | B | Displacement of (S)-4-(2,4-difluorophenyl-3-tritio) -4,5-dihydro-2-oxazolamine from human TAAR1 receptor expressed in HEK293 cells after 90 mins by beta counting analysis | Homo sapiens | 47 | cell-based format | Scientific Literature | ||
| 19. | ALA2213508 | F | Agonist activity at human TAAR1 receptor expressed in HEK293 cells after 30 mins | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 20. | ALA2215956 | F | Agonist activity at human TAAR1 receptor expressed in HEK293 cells after 30 mins relative to control | Homo sapiens | 6 | cell-based format | Scientific Literature |
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