| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA946280 | B | Inhibition of human JMJD2A by FDH coupled assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 2. | ALA1054738 | B | Inhibition of JMJD2A-mediated H3K9 demethylation activity at 3 mM | 5 | single protein format | Scientific Literature | |||
| 3. | ALA1055467 | B | Inhibition of JMJD2A-mediated H3K9 demethylation activity at 1 mM | 5 | single protein format | Scientific Literature | |||
| 4. | ALA1070284 | B | Inhibition of JMJD2A by MALDI-TOF assay | 11 | single protein format | Scientific Literature | |||
| 5. | ALA1219075 | B | Inhibition of recombinant His-tagged JMJD2A expressed in Escherichia coli Rosetta 2 (DE3) pLysS cells by formaldehyde dehydrogenase-coupled assay | 15 | cell-based format | Scientific Literature | |||
| 6. | ALA1738626 | B | PUBCHEM_BIOASSAY: JMJD2A counterscreen for GASC1 inhibitors Measured in Biochemical System Using Plate Reader - 2043-02_Inhibitor_Dose_CherryPick_Activity. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2123] | Homo sapiens | 52 | biochemical format | PubChem BioAssays | ||
| 7. | ALA1737991 | F | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of JMJD2A-Tudor Domain. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504402] | Homo sapiens | 51,376 | assay format | PubChem BioAssays | ||
| 8. | ALA1942535 | B | Inhibition of KDM4A | 8 | single protein format | Scientific Literature | |||
| 9. | ALA1942545 | B | Ratio of DMOG IC50 to compound IC50 for KDM4A | 1 | single protein format | Scientific Literature | |||
| 10. | ALA2173248 | B | Inhibition of JMJD2A | 1 | single protein format | Scientific Literature | |||
| 11. | ALA2173263 | B | Inhibition of JMJD2A catalytic domain by mass spectrophotometric analysis | 1 | single protein format | Scientific Literature | |||
| 12. | ALA2389133 | B | Inhibition of JMJD2A tudor domain (unknown origin) using histone H4 peptide trimethylated on lysine 20 as substrate | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA2395585 | B | Binding affinity to JMJD2A (unknown origin) up to 10 uM by fluorescence polarization assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA2396332 | B | Inhibition of JMJD2A (unknown origin) | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 15. | ALA2427609 | B | Inhibition of KDM4A (unknown origin) using H3K9me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assay | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 16. | ALA3390926 | B | Inhibition of Flag-tagged JMJD2A in human HeLa cells using H3K9me3 peptide as substrate by immunofluorescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA3390933 | B | Inhibition of JMJD2A (unknown origin) using ARK(me3)STGGK peptide as substrate preincubated for 1 to 30 mins followed by substrate addition by MALDI-TOF/MS analysis | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 18. | ALA3363696 | B | Inhibition of recombinant human KDM4A (1 to 347 aa) expressed in Escherichia coli using calf thymus histone H3 as substrate after 30 mins by Western blotting | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA3363698 | B | Inhibition of recombinant human KDM4A (1 to 347 aa) expressed in Escherichia coli using H3K9me3 peptide as substrate assessed as residual activity after 30 mins by FDH-coupled assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA3363700 | B | Competitive inhibition of recombinant human KDM4A (1 to 347 aa) expressed in Escherichia coli using H3K9me3 peptide as substrate after 30 mins by double-reciprocal plot method | Homo sapiens | 1 | assay format | Scientific Literature |
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