# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA995017 | B | Inhibition of RIOK2 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
2. | ALA1052945 | B | Inhibition of RIOK2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
3. | ALA1066098 | B | Inhibition of RIOK2 at 10 uM | 2 | ALA1152632 | single protein format | Scientific Literature | ||
4. | ALA1166841 | B | Inhibition of RIOK2 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
5. | ALA1175251 | B | Inhibition of RIOK2 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
6. | ALA1244956 | B | Binding affinity to RIOK2 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
7. | ALA1827240 | B | Activity of RIOK2 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
8. | ALA1908808 | B | Binding constant for RIOK2 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
9. | ALA2020366 | B | Inhibition of RIOK2 at 10 uM relative to control | 1 | ALA2016464 | single protein format | Scientific Literature | ||
10. | ALA2212013 | B | Inhibition of RIOK2 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
11. | ALA2214440 | B | Inhibition of RIOK2 | 1 | ALA2203257 | single protein format | Scientific Literature | ||
12. | ALA2215616 | B | Binding affinity to T7-phage-tagged RIOK2 by PCR analysis | 1 | ALA2203077 | single protein format | Scientific Literature | ||
13. | ALA2396460 | B | Competitive binding affinity to RIOK2 (unknown origin) assessed as enzyme remaining bound to anchored active-site ligand at 10 uM relative to control | Homo sapiens | 1 | ALA2390846 | single protein format | Scientific Literature | |
14. | ALA3366584 | B | Inhibition of RIOK2 (unknown origin) assessed as residual activity at 10 uM relative to control | Homo sapiens | 1 | ALA3352819 | single protein format | Scientific Literature | |
15. | ALA3430833 | B | Delta TM value showing the stabilisation of RIOK2 produced by compound binding | Homo sapiens | 156 | ALA1145498 | single protein format | Scientific Literature | |
16. | ALA3626280 | B | Inhibition of RIOK2 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3621137 | single protein format | Scientific Literature | |
17. | ALA3631579 | B | Inhibition of RIOK2 (unknown origin) assessed as remaining activity at 10 uM by high-throughput assay relative to control | Homo sapiens | 1 | ALA3627674 | single protein format | Scientific Literature | |
18. | ALA3734228 | B | Inhibition of N-terminal GST-fused full length human recombinant RIOK2 expressed in baculovirus Sf21 cells assessed as reduction in kinase auto-phosphorylation at 1 uM in presence of ATP incubated for 1 hr by ELISA method | Homo sapiens | 38 | ALA3727348 | cell-based format | Patent Bioactivity Data | |
19. | ALA3734229 | B | Inhibition of N-terminal GST-fused full length human recombinant RIOK2 expressed in baculovirus Sf21 cells assessed as reduction in kinase auto-phosphorylation at 10 uM in presence of ATP incubated for 1 hr by ELISA method | Homo sapiens | 41 | ALA3727348 | cell-based format | Patent Bioactivity Data | |
20. | ALA3771953 | B | Inhibition of human recombinant RIOK2 assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3769377 | single protein format | Scientific Literature |