| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA981786 | B | Inhibition of ULK1 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 2. | ALA1021462 | B | Inhibition of ULK1 assessed as enzyme activity relative to control | 1 | ALA1151738 | single protein format | Scientific Literature | ||
| 3. | ALA1059394 | B | Inhibition of ULK1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 4. | ALA1168303 | B | Inhibition of ULK1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
| 5. | ALA1175114 | B | Inhibition of ULK1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 6. | ALA1245019 | B | Binding affinity to ULK1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 7. | ALA1679293 | B | Binding affinity to ULK1 at 10 uM by immobilized ligand displacement assay | 1 | ALA1671850 | single protein format | Scientific Literature | ||
| 8. | ALA1826219 | B | Activity of ULK1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 9. | ALA1908613 | B | Binding constant for ULK1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 10. | ALA1944388 | B | Inhibition of ULK1 at 1 uM | 1 | ALA1938300 | single protein format | Scientific Literature | ||
| 11. | ALA2154990 | B | Binding affinity to ULK1 | 1 | ALA2150858 | single protein format | Scientific Literature | ||
| 12. | ALA2209239 | B | Inhibition of ULK2 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
| 13. | ALA3388694 | B | Inhibition of ULK1 (unknown origin) assessed as remaining enzyme activity at 10 uM by radioactive [33P]-ATP filter binding assay | Homo sapiens | 1 | ALA3351385 | single protein format | Scientific Literature | |
| 14. | ALA3606871 | B | Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubated for 7 mins | Homo sapiens | 5 | ALA3603808 | cell-based format | Scientific Literature | |
| 15. | ALA3626294 | B | Inhibition of ULK1 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3621137 | single protein format | Scientific Literature | |
| 16. | ALA3631618 | B | Inhibition of ULK1 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
| 17. | ALA3750199 | B | Inhibition of human ULK1 using MBP substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
| 18. | ALA3816874 | B | Inhibition of human ULK1 at 1 uM using MBP substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
| 19. | ALA3991921 | B | Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry. | Homo sapiens | 235 | ALA3991601 | subcellular format | Kuster lab chemical proteomics drug profiling | |
| 20. | ALA3995069 | B | Inhibition of human ULK1 (M1 to T309 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by KINOMEscan assay relative to control | Homo sapiens | 1 | ALA3994581 | assay format | Scientific Literature |
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