| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA691189 | F | In vitro agonist potency was evaluated in HEK293 cells transfected with human melanocortin receptor (hMC4R) | 25 | ALA1136147 | cell-based format | Scientific Literature | ||
| 2. | ALA708681 | F | Effective concentration for cAMP accumulation relative to alpha-MSH at human MC4R | 1 | ALA1136492 | assay format | Scientific Literature | ||
| 3. | ALA710020 | B | Binding affinity towards MCR-4 receptor | 1 | ALA1135101 | single protein format | Scientific Literature | ||
| 4. | ALA712741 | F | Maximum percent cAMP accumulation at 10 uM relative to alpha-MSH at Melanocortin-4 receptor | Homo sapiens | 7 | ALA1135618 | assay format | Scientific Literature | |
| 5. | ALA878334 | B | Binding affinity against human Melanocortin-4 receptor | Homo sapiens | 2 | ALA1135658 | single protein format | Scientific Literature | |
| 6. | ALA712742 | B | Inhibition of binding to human Melanocortin-4 receptor (hMC4R) | Homo sapiens | 12 | ALA1135991 | single protein format | Scientific Literature | |
| 7. | ALA712743 | B | Evaluated for Functional Activity at Melanocortin-4 receptor as effective concentration at 50% maximum CMP accumulation | 1 | ALA1135618 | single protein format | Scientific Literature | ||
| 8. | ALA884503 | F | Evaluated for Functional Activity at Melanocortin-4 receptor as effective concentration at 50% maximum CMP accumulation | 5 | ALA1135618 | assay format | Scientific Literature | ||
| 9. | ALA712744 | F | Functional activity as concentration at 50% maximum cAMP accumulation in human Melanocortin-4 receptor | 1 | ALA1135618 | assay format | Scientific Literature | ||
| 10. | ALA712745 | B | Binding affinity against human Melanocortin-4 receptor | Homo sapiens | 11 | ALA1135658 | single protein format | Scientific Literature | |
| 11. | ALA712746 | B | Binding affinity against human Melanocortin-4 receptor | Homo sapiens | 1 | ALA1135658 | single protein format | Scientific Literature | |
| 12. | ALA712747 | B | Evaluated for binding affinity against Melanocortin-4 receptor by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cells | 8 | ALA1135618 | cell-based format | Scientific Literature | ||
| 13. | ALA712748 | B | Evaluated for binding affinity against human Melanocortin-4 receptor (hMC4R) by displacing [125I]NDP-alpha-MSH radioligand expressed in CHO cells | 1 | ALA1135618 | cell-based format | Scientific Literature | ||
| 14. | ALA712906 | B | Binding affinity for human Melanocortin-4 receptor (hMC4R) | Homo sapiens | 12 | ALA1135991 | single protein format | Scientific Literature | |
| 15. | ALA712907 | F | Stimulation of intracellular cAMP levels in CHO cells expressing human Melanocortin-4 receptor | Homo sapiens | 12 | ALA1135991 | cell-based format | Scientific Literature | |
| 16. | ALA712908 | F | Percentage of cAMP accumulation at 10 uM relative to alpha-MSH at human Melanocortin-4 receptor | 1 | ALA1135618 | assay format | Scientific Literature | ||
| 17. | ALA714366 | F | Agonist activity against human Melanocortin-4 receptor | Homo sapiens | 3 | ALA1135658 | assay format | Scientific Literature | |
| 18. | ALA878339 | F | Agonist potency at human Melanocortin-4 receptor | Homo sapiens | 7 | ALA1135658 | assay format | Scientific Literature | |
| 19. | ALA714367 | F | Agonist potency at human Melanocortin-4 receptor | Homo sapiens | 1 | ALA1135658 | assay format | Scientific Literature | |
| 20. | ALA714368 | B | pA2 value for human Melanocortin-4 receptor | Homo sapiens | 10 | ALA1135658 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!