# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1035863 | B | Binding affinity to human ACTR2 at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
2. | ALA3991611 | B | Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry. | Homo sapiens | 223 | ALA3991601 | subcellular format | Kuster lab chemical proteomics drug profiling | |
3. | ALA4055144 | B | Inhibition of ACTR2 (unknown origin) assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | single protein format | Scientific Literature | |
4. | ALA4118563 | B | Binding affinity to ACTR2 in human NCI-H23 cells at 1 uM by mass spectrometry based pull down assay | Homo sapiens | 1 | ALA4118021 | cell-based format | Scientific Literature | |
5. | ALA4118811 | B | Binding affinity to ACTR2 in human NCI-H358 cells at 1 uM by mass spectrometry based pull down assay | Homo sapiens | 1 | ALA4118021 | cell-based format | Scientific Literature | |
6. | ALA4379133 | B | Inhibition of human recombinant ACTR2 (162 to end residues) using casein as substrate incubated for 120 mins in presence of [gamma-33P]ATP by radiometric scintillation counting analysis | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
7. | ALA4728245 | B | Binding affinity to ACTR2 (unknown origin) assessed as change in melting temperature at 10 uM incubated for 10 mins using SYPRO orange dye by RT-PCR-based fluorescence assay | Homo sapiens | 1 | ALA4725345 | single protein format | Scientific Literature | |
8. | ALA4880946 | B | ACTR2(h) Eurofins Kinase panel | Homo sapiens | 1 | ALA4507268 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
9. | ALA4884211 | B | ACTR2(h) Eurofins kinase panel | Homo sapiens | 1 | ALA4507319 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
10. | ALA4887766 | B | ACTR2(h) Millipore kinase panel | Homo sapiens | 1 | ALA4800729 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
11. | ALA5059015 | B | ACTR2(h) Kinase panel | Homo sapiens | 1 | ALA5058645 | single protein format | Donated Chemical Probes - SGC Frankfurt |