| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA995027 | B | Inhibition of PFTK1 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 2. | ALA1051350 | B | Binding constant for full-length PFTK1 | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 3. | ALA1057582 | B | Inhibition of PFTK1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 4. | ALA1166616 | B | Inhibition of PFTK1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
| 5. | ALA1175194 | B | Inhibition of PFTK1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 6. | ALA1244562 | B | Binding affinity to PFTK1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 7. | ALA1827564 | B | Activity of PFTK1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 8. | ALA1908767 | B | Binding constant for PFTK1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 9. | ALA1942459 | B | Inhibition of human PFTAIRE1 in HL-60 cells lysate assessed as reduction of labeling of acyl-phosphate ATP probe at 100 nM | Homo sapiens | 4 | ALA1938230 | cell-based format | Scientific Literature | |
| 10. | ALA2214969 | B | Inhibition of PFTK1 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
| 11. | ALA2424038 | B | Inhibition of PFTAIRE1 in human PC3 cell lysates at 10 uM using desthiobiotin-tagged ATP probe AX9989 followed by trypsinization by LC/MS analysis | Homo sapiens | 12 | ALA2417377 | single protein format | Scientific Literature | |
| 12. | ALA2429140 | B | Competitive binding affinity to PFTK1 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | ALA2424622 | single protein format | Scientific Literature | |
| 13. | ALA3111953 | B | Inhibition of PFTK1 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
| 14. | ALA3631904 | B | Inhibition of PFTK1 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
| 15. | ALA4025301 | B | Inhibition of wild-type human full length PFTK1 (M1 to H451 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
| 16. | ALA4034451 | B | Inhibition of PFTAIRE1 Lysine 1 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
| 17. | ALA4034452 | B | Inhibition of PFTAIRE1 Lysine 2 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
| 18. | ALA4044112 | B | Inhibition of wild-type human full length PFTK1 (M1 to H451 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | assay format | Scientific Literature | |
| 19. | ALA4045795 | B | Inhibition of PFTAIRE1 conserved Lys1 (LVALKVIR) in human PBMC at 1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature | |
| 20. | ALA4046036 | B | Inhibition of PFTAIRE1 conserved Lys1 (LVALKVIR) in human PBMC at 0.1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!