# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA982813 | B | Inhibition of histidine-tagged recombinant tankyrase-1 by flashplate scintillation proximity assay | 1 | ALA1140140 | single protein format | Scientific Literature | ||
2. | ALA1060809 | B | Inhibition of human tankyrase 1 catalytic domain expressed in Escherichia coli up to 500 nM | Homo sapiens | 2 | ALA1153049 | assay format | Scientific Literature | |
3. | ALA1074657 | B | Inhibition of Tankyrase 1 | 2 | ALA1153250 | single protein format | Scientific Literature | ||
4. | ALA1116320 | B | Inhibition of human TANK1 C-terminal domain by trichloroacetic acid precipitation assay | Homo sapiens | 1 | ALA1157008 | single protein format | Scientific Literature | |
5. | ALA1119030 | B | Inhibition of TNKS1 | 1 | ALA1155445 | single protein format | Scientific Literature | ||
6. | ALA1119032 | B | Binding affinity to TNKS1 | 1 | ALA1155445 | single protein format | Scientific Literature | ||
7. | ALA1119038 | B | Binding affinity to human recombinant TNSK1 expressed in Escherichia coli by isothermal titration calorimetry | Homo sapiens | 1 | ALA1155445 | assay format | Scientific Literature | |
8. | ALA2020820 | B | Inhibition of GST-tagged TNKS1P catalytic domain autoPARsylation measuring nicotinamide concentration after 2 hrs by LC-MS analysis | 6 | ALA2016557 | single protein format | Scientific Literature | ||
9. | ALA2020827 | B | Binding affinity to biotinylated Avi-tagged TNKS1 | 1 | ALA2016557 | single protein format | Scientific Literature | ||
10. | ALA2034621 | B | Inhibition of TNKS1 | 2 | ALA2029260 | single protein format | Scientific Literature | ||
11. | ALA2317531 | B | Inhibition of N-terminal His6-tagged human TNKS1 (1091 to 1325 amino acid residues) after 60 mins by autoparsylation assay | Homo sapiens | 4 | ALA2311538 | single protein format | Scientific Literature | |
12. | ALA2330786 | B | Inhibition of TNSK1 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assay | Homo sapiens | 1 | ALA2321812 | single protein format | Scientific Literature | |
13. | ALA2341188 | B | Inhibition of human 6XHis-tagged TNKS1 SAM-ART domain (1030 to 1317 amino acid residues) by fluorescence assay | Homo sapiens | 10 | ALA2331472 | single protein format | Scientific Literature | |
14. | ALA2382486 | B | Inhibition of TNKS1 (unknown origin) | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
15. | ALA2384487 | B | Inhibition of 6XHis-tagged tankyrase1 (1091 to 1325) (unknown origin) after 60 mins in presence of NAD | Homo sapiens | 32 | ALA2380263 | single protein format | Scientific Literature | |
16. | ALA2422482 | B | Inhibition of TNSK1 (unknown origin) assessed as nicotinamide concentration by LC-MS analysis | Homo sapiens | 6 | ALA2417384 | single protein format | Scientific Literature | |
17. | ALA2428877 | B | Inhibition of N-terminal GST-tagged human TNKS1 expressed in baculovirus infected sf21 cells after 60 mins by LC-MS analysis | Homo sapiens | 8 | ALA2424545 | cell-based format | Scientific Literature | |
18. | ALA2433652 | B | Inhibition of human TNKS1 (1030 to 1317) using NAD+ as substrate by fluorescence assay | Homo sapiens | 32 | ALA2429767 | single protein format | Scientific Literature | |
19. | ALA3102115 | B | Inhibition of human tankyrase1 after 30 mins by spectrophotometry | Homo sapiens | 13 | ALA3098040 | single protein format | Scientific Literature | |
20. | ALA3102117 | B | Inhibition of tankyrase1 (unknown origin) | Homo sapiens | 1 | ALA3098040 | single protein format | Scientific Literature |