# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA962978 | B | Inhibition of recombinant BAT5 transfected in HEK293T cells by SDS-PAGE using rhodamine-tagged FP probe | 2 | ALA1151781 | cell-based format | Scientific Literature | ||
2. | ALA2209087 | B | Inhibition of BAT5 binding to FP-biotin in [12C][14N]-lysine, arginine and [13C6][15N2]-lysine, arginine labeled HEK293T cells at 20 uM after 1 hr by isotopic activity-based protein profiling-MudPIT assay | Homo sapiens | 1 | ALA2203175 | cell-based format | Scientific Literature | |
3. | ALA4330036 | B | Inhibition of ABHD16A (unknown origin) | Homo sapiens | 4 | ALA4325934 | single protein format | Scientific Literature | |
4. | ALA4330037 | B | Potency index, ratio of tetrahydrolipstatin IC50 to compound IC50 for inhibition of ABHD16A (unknown origin) | Homo sapiens | 3 | ALA4325934 | single protein format | Scientific Literature | |
5. | ALA4330038 | B | Inhibition of human ABHD16A expressed in HEK293 cells assessed as residual activity at 10 uM preincubated for 30 mins followed by 1-LG substrate addition and measured after 90 to 120 mins by fluorometric assay relative to control | Homo sapiens | 20 | ALA4325934 | cell-based format | Scientific Literature | |
6. | ALA4330040 | B | Inhibition of human ABHD16A expressed in HEK293 cells preincubated for 30 mins followed by 1-LG substrate addition and measured after 90 to 120 mins by fluorometric assay | Homo sapiens | 3 | ALA4325934 | cell-based format | Scientific Literature | |
7. | ALA4330041 | B | Reversible inhibition of human ABHD16A expressed in HEK293 cells preincubated for 30 mins followed by 40 fold compound dilution and subsequent 1-LG substrate addition and measured at 30 mins time interval for 120 mins by fluorometric assay | Homo sapiens | 3 | ALA4325934 | cell-based format | Scientific Literature | |
8. | ALA4330042 | B | Inhibition of human ABHD16A expressed in HEK293 cells assessed as residual activity at 100 uM preincubated for 30 mins followed by 1-LG substrate addition and measured after 90 to 120 mins by fluorometric assay relative to control | Homo sapiens | 2 | ALA4325934 | cell-based format | Scientific Literature | |
9. | ALA4330043 | B | Ratio of IC50 for reversible inhibition of human ABHD16A expressed in HEK293 cells to IC50 for inhibition of human ABHD16A expressed in HEK293 cells | Homo sapiens | 3 | ALA4325934 | cell-based format | Scientific Literature | |
10. | ALA4330050 | B | Inhibition of TAMRA-FP binding to human ABHD16A expressed in HEK293 cells at 20 to 200 uM preincubated for 1 hr followed by TAMRA-FP addition measured after 1 hr by fluorescence based ABPP analysis | Homo sapiens | 1 | ALA4325934 | cell-based format | Scientific Literature |