# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1032240 | B | Inhibition of ACVR2A at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
2. | ALA1060234 | B | Binding constant for ACVR2A kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
3. | ALA1057562 | B | Inhibition of ACVR2A assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
4. | ALA1168584 | B | Inhibition of ACVR2A at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
5. | ALA1174058 | B | Inhibition of ACVR2A at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
6. | ALA1244714 | B | Binding affinity to ACVR2A | 7 | ALA1240346 | single protein format | Scientific Literature | ||
7. | ALA1827637 | B | Activity of ACVR2A kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
8. | ALA1908535 | B | Binding constant for ACVR2A kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
9. | ALA2216366 | B | Inhibition of ACVR2A | 1 | ALA2203257 | single protein format | Scientific Literature | ||
10. | ALA2212085 | B | Inhibition of ACVR2A assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
11. | ALA2428335 | B | Competitive binding affinity to ACVR2A (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 4 | ALA2424622 | single protein format | Scientific Literature | |
12. | ALA3112124 | B | Inhibition of AVR2A (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
13. | ALA4025001 | B | Inhibition of wild-type human ACVR2A (V171 to T499 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
14. | ALA4043812 | B | Inhibition of wild-type human ACVR2A (V171 to T499 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | assay format | Scientific Literature | |
15. | ALA4153868 | B | Inhibition of ACVR2A (unknown origin) at 10 uM by [33P]-ATP radiometric assay | Homo sapiens | 6 | ALA4152228 | single protein format | Scientific Literature | |
16. | ALA4156891 | B | Binding affinity to wild-type human ACVR2A (V171 to T499 residues) expressed in bacterial expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
17. | ALA4185670 | B | Binding affinity to wild-type human ACVR2A (V171 to T499 residues) expressed in Escherichia coli BL21 at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | assay format | Scientific Literature | |
18. | ALA4190854 | B | Inhibition of recombinant human ACTR2 (162 to end residues) at 1 uM using casein as substrate after 120 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4190187 | single protein format | Scientific Literature | |
19. | ALA4230570 | B | Binding affinity to wild-type human ACVR2A (V171 to T499 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
20. | ALA4263987 | B | Inhibition of full length GST-tagged human ACVR2A expressed in Baculovirus expression system by LanthaScreen assay | Homo sapiens | 1 | ALA4261595 | assay format | Scientific Literature |