# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1000438 | B | Inhibition of human DLK expressed in baculovirus insect cell system | Homo sapiens | 3 | ALA1140055 | assay format | Scientific Literature | |
2. | ALA1034101 | B | Inhibition of DLK at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
3. | ALA1055292 | B | Inhibition of DLK assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
4. | ALA1114872 | B | Inhibition of DLK at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
5. | ALA1168855 | B | Inhibition of DLK at 1 uM | 8 | ALA1165965 | single protein format | Scientific Literature | ||
6. | ALA1174317 | B | Inhibition of DLK at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
7. | ALA1244793 | B | Binding affinity to DLK | 7 | ALA1240346 | single protein format | Scientific Literature | ||
8. | ALA1826205 | B | Activity of DLK kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
9. | ALA2216440 | B | Inhibition of DLK assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
10. | ALA2344392 | B | Inhibition of DLK (unknown origin) | Homo sapiens | 1 | ALA2331331 | single protein format | Scientific Literature | |
11. | ALA2428158 | B | Competitive binding affinity to DLK (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | ALA2424622 | single protein format | Scientific Literature | |
12. | ALA2439120 | B | Binding affinity to human wild type DLK by qPCR analysis | Homo sapiens | 1 | ALA2434948 | single protein format | Scientific Literature | |
13. | ALA2439122 | B | Inhibition of human wild type DLK at 1 uM by qPCR analysis relative to control | Homo sapiens | 1 | ALA2434948 | single protein format | Scientific Literature | |
14. | ALA2439773 | B | Inhibition of human wild type DLK by qPCR analysis | Homo sapiens | 1 | ALA2434948 | single protein format | Scientific Literature | |
15. | ALA3377246 | B | Inhibition of DLK (unknown origin) by RT-FRET assay | Homo sapiens | 4 | ALA3351401 | single protein format | Scientific Literature | |
16. | ALA3630347 | B | Inhibition of DLK (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
17. | ALA4025092 | B | Inhibition of wild-type human full length DLK (M1 to P859 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
18. | ALA4043903 | B | Inhibition of wild-type human full length DLK (M1 to P859 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature | |
19. | ALA4054939 | B | Inhibition of wild-type human full length DLK (M1 to P859 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
20. | ALA4156982 | B | Binding affinity to wild-type human full length DLK (M1 to P859 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature |