# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1062872 | Binding | Binding constant for SRMS kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
2. | ALA1045666 | Binding | Binding affinity to SRMS assessed as percentage of kinase remaining bound to the bead at 1 uM by T7 phage display based binding assay | 1 | ALA1154183 | single protein format | Scientific Literature | ||
3. | ALA1052970 | Binding | Inhibition of SRMS assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
4. | ALA981777 | Binding | Inhibition of SRMS at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
5. | ALA1167705 | Binding | Inhibition of SRMS at 1 uM | 8 | ALA1165965 | single protein format | Scientific Literature | ||
6. | ALA1175019 | Binding | Inhibition of SRMS at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
7. | ALA1244293 | Binding | Inhibition of SRMS at 1 uM after 60 mins by FRET assay in presence of 100 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
8. | ALA1244983 | Binding | Binding affinity to SRMS | 7 | ALA1240346 | single protein format | Scientific Literature | ||
9. | ALA1251693 | Binding | Inhibition of SRMS at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature | ||
10. | ALA1826704 | Binding | Activity of SRMS kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
11. | ALA1827048 | Binding | Inhibition of SRMS at 1 uM | 3 | ALA1821716 | single protein format | Scientific Literature | ||
12. | ALA1908407 | Binding | Binding constant for SRMS kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
13. | ALA4387362 | Binding | Inhibition of recombinant full length human GST-tagged SRM expressed in baculovirus expression system at 0.1 uM using tyrosine-1 peptide as substrate incubated for 60 mins by Z'-LYTE assay relative to control | Homo sapiens | 2 | ALA4385643 | assay format | Scientific Literature | |
14. | ALA4389489 | Binding | Inhibition of wild-type human partial length SRMS (L208 to P488 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
15. | ALA4389966 | Binding | Inhibition of wild-type human partial length SRMS (L208 to P488 residues) expressed in mammalian expression system at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
16. | ALA4382770 | Binding | Binding affinity to wild-type human partial length SRMS (L208 to P488 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4382192 | assay format | Scientific Literature | |
17. | ALA3369198 | Binding | Inhibition of Srm (unknown origin) at 100 nM | Homo sapiens | 1 | ALA3297705 | single protein format | Scientific Literature | |
18. | ALA4365976 | Binding | Inhibition of wild-type human partial length SRMS (L208 to P488 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature | |
19. | ALA4366594 | Binding | Inhibition of human SRMS at 100 nM using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4364276 | single protein format | Scientific Literature | |
20. | ALA4377911 | Binding | Inhibition of human SRMS at 1 uM by radiometric method relative to control | Homo sapiens | 1 | ALA4376814 | single protein format | Scientific Literature |