| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA993459 | B | Binding affinity to human ALK2 at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
| 2. | ALA1032238 | B | Inhibition of ACVR1 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 3. | ALA1063697 | B | Binding constant for ACVR1 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 4. | ALA1057560 | B | Inhibition of ACVR1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 5. | ALA1057561 | B | Inhibition of ACVR1B assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 6. | ALA1066599 | B | Residual activity of ACV-R1 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 7. | ALA1046505 | B | Residual activity of ACV-R1 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 8. | ALA1047771 | B | Residual activity of ACV-R1 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 9. | ALA1168582 | B | Inhibition of ACVR1 at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
| 10. | ALA1174056 | B | Inhibition of ACVR1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 11. | ALA1244712 | B | Binding affinity to ACVR1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 12. | ALA1799787 | B | Inhibition of ACVR1 at 1 uM | 2 | ALA1795227 | single protein format | Scientific Literature | ||
| 13. | ALA1827636 | B | Activity of ACVR1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 14. | ALA1908516 | B | Binding constant for ACVR1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 15. | ALA1963721 | F | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: ACVR1 | 346 | ALA1201862 | assay format | PubChem BioAssays | ||
| 16. | ALA2216364 | B | Inhibition of ACVR1 | 1 | ALA2203257 | single protein format | Scientific Literature | ||
| 17. | ALA2212088 | B | Inhibition of ACVR1 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
| 18. | ALA2390524 | B | Inhibition of ALK2 (unknown origin) | Homo sapiens | 11 | ALA2384981 | single protein format | Scientific Literature | |
| 19. | ALA2406116 | B | Inhibition of ACVR1 (unknown origin) at 10 uM relative to control | Homo sapiens | 1 | ALA2401733 | single protein format | Scientific Literature | |
| 20. | ALA2428337 | B | Competitive binding affinity to ACVR1 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 4 | ALA2424622 | single protein format | Scientific Literature |
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