# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3630924 | Binding | Inhibition of PKAcbeta (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
2. | ALA3748052 | Binding | Inhibition of human PKAcbeta using [KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
3. | ALA826977 | Binding | Inhibition of human Protein kinase A beta | Homo sapiens | 6 | ALA1138659 | single protein format | Scientific Literature | |
4. | ALA871550 | Binding | Inhibition of PKAbeta by HTRF kinase assay | Homo sapiens | 2 | ALA1149344 | single protein format | Scientific Literature | |
5. | ALA1166813 | Binding | Inhibition of PKAC-beta at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
6. | ALA1175221 | Binding | Inhibition of PKAC-beta at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
7. | ALA1244928 | Binding | Binding affinity to PKAC-beta | 7 | ALA1240346 | single protein format | Scientific Literature | ||
8. | ALA1249687 | Binding | Inhibition of human PKA activity at 10 uM by radiometric assay | Homo sapiens | 2 | ALA1240306 | single protein format | Scientific Literature | |
9. | ALA1768516 | Binding | Inhibition of PKA activity using neurogranin as a substrate in presence of 50 uM ATP by mass spectrometry | 5 | ALA1764955 | single protein format | Scientific Literature | ||
10. | ALA1826685 | Binding | Activity of PKAC-beta kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
11. | ALA4352008 | Binding | Inhibition of recombinant full-length human PKAC beta at 10 uM using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4350961 | single protein format | Scientific Literature | |
12. | ALA4352498 | Binding | Inhibition of human PKAcb at 10 uM using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 1 | ALA4350963 | single protein format | Scientific Literature | |
13. | ALA4358076 | Binding | Binding affinity to wild-type human full length PKAC-beta (M1 to F351 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4354843 | assay format | Scientific Literature | |
14. | ALA1908579 | Binding | Binding constant for PKAC-beta kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
15. | ALA1039274 | Binding | Binding constant for full-length PKAC-beta | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
16. | ALA1057597 | Binding | Inhibition of PKACbeta assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
17. | ALA971638 | Binding | Inhibition of PKA-B | 1 | ALA1140084 | single protein format | Scientific Literature | ||
18. | ALA1017907 | Binding | Inhibition of PKAC-beta assessed as enzyme activity relative to control | 1 | ALA1151738 | single protein format | Scientific Literature | ||
19. | ALA981745 | Binding | Inhibition of PKAC-beta at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
20. | ALA2015484 | Binding | Inhibition of PKACb (PRKACB) at 10 uM | 1 | ALA2010722 | single protein format | Scientific Literature |