# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3630913 | Binding | Inhibition of PASK (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
2. | ALA3721069 | Binding | Inhibition of purified human PASK expressed in insect cells using MBP protein substrate incubated for 10 mins before ATP addition and measured after 1 hr by kinase-Glo luminescent kinase assay | Homo sapiens | 2 | ALA3714757 | cell-based format | Patent Bioactivity Data | |
3. | ALA3721070 | Binding | Inhibition of N-terminal GST-tagged human recombinant PASK kinase domain (879 to 1323 residues) expressed in insect cells using MBP protein substrate incubated for 120 mins in presence of [33P]ATP by scintillation counting based radiochemical assay | Homo sapiens | 2 | ALA3714757 | cell-based format | Patent Bioactivity Data | |
4. | ALA3721071 | Binding | Inhibition of human recombinant PASK using Ulight-peptide substrate incubated for 2 hrs by TR-FRET assay | Homo sapiens | 2 | ALA3714757 | single protein format | Patent Bioactivity Data | |
5. | ALA3721072 | Binding | Inhibition of purified human PASK expressed in insect cells using MBP protein substrate incubated for 10 mins before ATP addition and measured after 1 hr by kinase-Glo luminescent kinase assay | Homo sapiens | 10 | ALA3714759 | cell-based format | Patent Bioactivity Data | |
6. | ALA3721073 | Binding | Inhibition of purified human PASK kinase domain expressed in insect cells using MBP protein substrate incubated for 10 mins before ATP addition and measured after 1 hr by kinase-Glo luminescent kinase assay | Homo sapiens | 20 | ALA3714759 | cell-based format | Patent Bioactivity Data | |
7. | ALA3721074 | Binding | Inhibition of N-terminal GST-tagged human recombinant PASK kinase domain (879 to 1323 residues) expressed in insect cells using MBP protein substrate incubated for 120 mins in presence of [33P]ATP by scintillation counting method | Homo sapiens | 37 | ALA3714759 | cell-based format | Patent Bioactivity Data | |
8. | ALA3721075 | Binding | Inhibition of human recombinant PASK kinase domain using Ulight-peptide substrate incubated for 2 hrs by TR-FRET assay | Homo sapiens | 4 | ALA3714759 | single protein format | Patent Bioactivity Data | |
9. | ALA3721077 | Binding | Inhibition of purified human PASK expressed in insect cells using MBP protein substrate incubated for 10 mins before ATP addition and measured after 1 hr by kinase-Glo luminescent kinase assay | Homo sapiens | 17 | ALA3714736 | cell-based format | Patent Bioactivity Data | |
10. | ALA3721078 | Binding | Inhibition of N-terminal GST-tagged human recombinant PASK kinase domain (879 to 1323 residues) expressed in insect cells using MBP protein substrate incubated for 120 mins in presence of [33P]ATP by scintillation counting based radiochemical assay | Homo sapiens | 57 | ALA3714736 | cell-based format | Patent Bioactivity Data | |
11. | ALA3721079 | Binding | Inhibition of human recombinant PASK using Ulight-peptide substrate incubated for 2 hrs by TR-FRET assay | Homo sapiens | 79 | ALA3714736 | single protein format | Patent Bioactivity Data | |
12. | ALA3720757 | Binding | Inhibition of N-terminal GST-tagged human recombinant PASK kinase domain (879 to 1323 residues) expressed in insect cells using MBP protein substrate incubated for 120 mins in presence of [33P]ATP by scintillation counting based radiochemical assay | Homo sapiens | 50 | ALA3714726 | cell-based format | Patent Bioactivity Data | |
13. | ALA3720795 | Binding | Inhibition of human recombinant PASK using Ulight-peptide substrate incubated for 2 hrs by TR-FRET assay | Homo sapiens | 146 | ALA3714726 | single protein format | Patent Bioactivity Data | |
14. | ALA3720804 | Binding | Inhibition of N-terminal GST-tagged human recombinant PASK kinase domain (879 to 1323 residues) expressed in insect cells using MBP protein substrate incubated for 120 mins in presence of [33P]ATP by scintillation counting based radiochemical assay | Homo sapiens | 8 | ALA3714765 | cell-based format | Patent Bioactivity Data | |
15. | ALA3720805 | Binding | Inhibition of human recombinant PASK using Ulight-peptide substrate incubated for 2 hrs by TR-FRET assay | Homo sapiens | 10 | ALA3714765 | single protein format | Patent Bioactivity Data | |
16. | ALA3720806 | Binding | Inhibition of purified human PASK expressed in insect cells using MBP protein substrate incubated for 10 mins before ATP addition and measured after 1 hr by kinase-Glo luminescent kinase assay | Homo sapiens | 4 | ALA3714765 | cell-based format | Patent Bioactivity Data | |
17. | ALA3720807 | Binding | Inhibition of V5-tagged wild type human PASK expressed HEK293T cells assessed as reduction in enzyme autophosphorylation incubated for 24 hrs by SDS-PAGE and Western blot method | Homo sapiens | 1 | ALA3714765 | cell-based format | Patent Bioactivity Data | |
18. | ALA3720972 | Binding | Inhibition of human recombinant PASK using Ulight-peptide substrate incubated for 2 hrs by TR-FRET assay | Homo sapiens | 23 | ALA3714735 | single protein format | Patent Bioactivity Data | |
19. | ALA3720973 | Binding | Inhibition of purified full-length human PASK expressed in insect cells using MBP protein substrate incubated for 10 mins before ATP addition and measured after 1 hr by kinase-Glo luminescent kinase assay | Homo sapiens | 50 | ALA3714729 | cell-based format | Patent Bioactivity Data | |
20. | ALA3720974 | Binding | Inhibition of purified human PASK kinase domain expressed in insect cells using MBP protein substrate incubated for 10 mins before ATP addition and measured after 1 hr by kinase-Glo luminescent kinase assay | Homo sapiens | 48 | ALA3714729 | cell-based format | Patent Bioactivity Data |